Noj qab haus huv, Npaj
"Elefloks": cov lus qhia rau kev siv, tiag tiag counterparts
"Elefloks" yog ib tug fluoroquinolone pab pawg neeg. Cov kev npaj muaj ib qho kev antimicrobial nyhuv. Lub ntsiab tshuaj tivthaiv - levofloxacin. Tshuaj thiab tshuaj "Elefloks" qhia nyob rau hauv daim tawv nqaij kab mob, mob dab nyob rau hauv nqaij mos mos, Septicemia, mob ntsws, prostatitis kab mob etiology, mob sinusitis nyob rau hauv lwm yam kab mob thiab kab mob xwm.
Muaj pes tsawg leeg thiab rau hauv daim ntawv ntawm "Elefloksa" tshuaj
Cov tshuaj no muaj nyob rau ob ntau npaum ntaub ntawv - cov ntsiav tshuaj (packing 5 thiab 10 pcs.), Tso dej tshuaj (100 ml flasks). Ib tug tov uas muaj 5 mg / ml ntawm active ingredient. Cov ntsiav tshuaj tej zaum yuav muaj li ntawm 250 los yog 500 mg ntawm lub ntsiab tivthaiv.
Muaj pes tsawg leeg ntawm lub ntsiav tshuaj muaj xws li ib co cam: polysorbate 80, magnesium stearate, crospovidone, hypromellose, MCC (Avicel PH 101, 102).
Tshuaj tua kab mob "Elefloks" nyob rau hauv daim ntawv ntawm cov ntsiav tshuaj coated ntsiav tshuaj, uas yog siv los tsim hlau oxide (daj, liab), macrogol, titanium dioxide. Ib tug tov raws li ib tug pab tivthaiv muaj sodium hydroxide, dej kev txhaj tshuaj, hydrochloric acid thiab anhydrous dextrose.
Pharmacological kev txiav txim "Elefloks" tshuaj
Active muaj depressing ntxim rau cov synthesis ntawm cov kab mob DNA. Morphological kev hloov tshwm sim uas cuam tshuam rau cytoplasm, membrane thiab cell phab ntsa ntawm kab mob ua rau lawv tuag. Cov dab muab ib tug bactericidal thiab antimicrobial los. Rau ib txhia tshuaj raug co thiab aerobic (gram-zoo, gram-tsis zoo), thiab lwm yam kab mob.
Nyob rau hauv qhov ncauj siv ntawm cov tshuaj "Elefloks" ib feem ntawm lub cuab tam yog sai absorbed los ntawm tus mob huam yuav luag tag. Thaum ib tug ntau npaum ntawm 500 mg active ingredient bioavailability yog yuav luag 100 feem pua, nrog rau cov ntshav thwj toob ntawm - ib tug nruab nrab ntawm 35 feem pua. Cov tshuaj penetrates zoo nyob rau hauv ib co ntaub so ntswg thiab kabmob. Ib tug me ib feem yog oxidized deacetylated los ntawm lub siab. Mas nyob rau hauv lub tshem tawm ntawm cov tshuaj los ntawm lub cev uas muaj ob lub raum.
Indications "Elefloks" npaj
"Elefloks" analogues yog siv nyob rau hauv daim tawv nqaij qhov chaw mob, prostatitis, ib tug kab mob uas muaj feem xyuam rau cov pa ib ntsuj av tau, cov kabmob uas ua tau lub urinary system. Lub medicament yog siv raws li ib tug adjunct kho nrog tuberculosis, uas nws lub cev yog txhais raws li ruaj khov.
Tshuaj kho cov kab thiab inflammatory kab mob tshwm sim los ntawm qhov tsis zoo feem ntawm kab mob differing rhiab heev rau levofloxacin. "Elefloks" qhia ntawv nyob rau daim ntawv thov tso cai rau koj mus muab thaum pom:
- prostatitis yog ib tug kab mob etiology;
- sinusitis nyob rau hauv mob daim ntawv;
- intra-plab kab mob;
- ntev bronchitis sharpened zoo lawm;
- kab dab nyob rau hauv lub mob txeeb zig nrog los sis tsis muaj teeb meem;
- kab mob rau ntawm daim tawv nqaij thiab nqaij mos mos;
- lub zej lub zos-kis tau mob ntsws;
- kab mob uas muaj feem xyuam rau Upper pa kabmob;
- Septicemia;
- mob;
- tuberculosis resistant mus rau lub kev txiav txim ntawm cov tshuaj (los "Elefloksa" yog ua los ntawm kev siv txoj kev kho).
Contraindications tau txais "Elefloks" tshuaj
Rau cov tshuaj muaj ib tug xov tooj ntawm contraindications. "Elefloks" cov lus qhia rau kev siv tsis pub siv nyob rau hauv qaug dabpeg, convulsive mob, tus me nyuam-tau cov kabmob thiab lactation. Cov tshuaj muab rau ib tug neeg mob, uas nws muaj hnub nyoog yog tsawg tshaj li 18 xyoo. Contraindications xws li txog leeg raug mob, uas ua uas siv quinolones txoj kev kho, thiab muaj zog xob cov Cheebtsam ntawm cov txhais tau tias. Yog li ntawd, ua ntej koj ua ntawv thov yuav tsum tau ua tib zoo kawm txog yeeb tshuaj thiab tham ib tug tshwj xeeb.
Thaum lub sij hawm ntawm kev kho mob yuav tsum tau tshwj xeeb mloog mus rau tus neeg mob rau kev ua txhaum nyob rau hauv lub chaw ua hauj lwm ntawm ob lub raum, tsis muaj peev xwm ntawm glucose-6-phosphate dehydrogenase. Thaum lub sij hawm kev kho mob ntawm cov neeg laus cov neeg mob yuav tsum tau kho mob saib xyuas.
Txoj kev siv "Elefloks" tshuaj
"Elefloks" analogues yog pom zoo kom siv thaum muaj mov noj los yog nyob rau hauv pem hauv ntej ntawm lawv (30 feeb ua ntej noj mov). Cov ntsiav tshuaj yuav npaum li cas tsuas yog raws li ib tug tag nrho daim ntawv nrog ib tug txaus tus nqi ntawm cov dej sov so.
Yeej, ntawm thawj zaug rau theem ntawm kev kho mob txhua txhua hnub tshuaj noj mus rau hauv kev ua raws cai nrog lub luv ntawm 1-2 xuab moos. Cov tshuaj nyob ntawm tus kab mob no, cov heev thiab cov hoob kawm ntawm nws rhiab heev rau cov tshuaj yav kab mob.
Feem ntau, thaum creatinine clearance siab tshaj 50 mL / min, xws kiag thov:
- teeb meem ntawm mob ntsws - ib koob tshuaj ib hnub twg - 250-500 mg, ib chav kawm ntev los ntawm ib lub lim tiam mus rau kaum hnub;
- ntws mob sinusitis - tshuaj "Elefloks" (500 mg) yog coj txhua txhua hnub rau kaum hnub los yog ob lub lis piam;
- lub zej lub zos-kis tau mob ntsws - siv 1000 mg ntawm yeeb tshuaj ib hnub twg nyob rau hauv 2 faib koob tshuaj rau 1-2 lub lis piam;
- nyuab los ntawm tus kab mob, rau lub mob txeeb zig - txhua hnub koob tshuaj sau raws nkaus Ii 250 mg ntawm cov tshuaj, cov kev ntev yog ib tug me ntsis ntau tshaj ib lub lim tiam, cov kev kho mob yog ntev, yog tias tsim nyog;
- pathology, uas muaj feem xyuam rau cov mob txeeb zig, thiab muaj cov tsis muaj teeb meem - txog 4 hnub twb txais yuav los ntawm 250 mg ntawm cov tshuaj;
- prostatitis tshwm sim los ntawm cov kab mob, - yuav tsum tau ntev-lub sij hawm kev kho mob, tej zaum tsis pub dhau 28 hnub los ntawm 500 mg "Elefloksa" txhua hnub;
- sinusitis - Kho tsim ntsiav tshuaj nyob rau hauv ib tug txhua txhua hnub koob tshuaj ntawm 500 mg;
- intraabdominal kab mob - koob tshuaj rau txhua txhua hnub saib xyuas yog 500 mg, hauv chav kawm ntev nyob rau hauv lub complex kev kho mob - 1-2 lub lis piam;
- cov kab mob nyob rau hauv uas lub qhov cov tawv nqaij thiab nqaij mos - yuav tsum tau kho nrog ib tug muab ob npaug rau tau txais 250 mg los yog 500 mg tshuaj txhua txhua hnub rau ob lub lim piam;
- tuberculosis resistant mus rau lub kev txiav txim ntawm lwm yam tshuaj - rau txoj kev kho mob yog tsim nyog los noj txhua txhua hnub rau 500 mg ntawm yeeb tshuaj (muaj peev xwm txais tau 2-fold) rau peb lub hlis.
Cov neeg mob uas mob raum nyob rau hauv tej yam muaj nuj nqis QC (ml / min) "Elefloks" cov lus qhia rau kev siv yuav tau txais raws li nram no:
- QC 50-20 - thawj noj 250 mg, thiab tom qab ntawd - 125-250 mg (tejzaum nws phua rau hauv ob peb lub sij hawm);
- QC 10-19 - thawj tau txais 500 mg ib hnub twg, nrog ntxiv kev kho mob - 125 mg rau ib 12-48 teev;
- CC hauv qab no 10 - txhua leej txhua tus yog ua tib yam li nyob rau hauv lub yav dhau los cov ntaub ntawv, tab sis cov tshuaj no yog siv ntau tshaj li ib zaug nyob rau hauv 12-48 teev, thiab txhua txhua 1-2 hnub.
Ua los ntawm cov tshuaj "Elefloks" dropper muab tso rau yam tsawg ib teev. Ntxiv kev kho mob nyob rau hauv tus neeg mob tus mob. Ib tug kev hloov mus rau lub ntsiav tshuaj mus rau lub ntau npaum, uas muab tso rau ib tug dropper. Nyob rau hauv cov mob uas tib neeg lub cev yog raug rau peritoneal lim ntshav thiab hemodialysis muab ntxiv koob tshuaj medicament yog yuav tsum tau.
Kev kho mob ntawm cov neeg laus cov neeg mob uas muaj teeb meem siab, nqa tawm rau 48-72 teev los yog ntev dua, kom txog rau thaum cov tsos mob ploj, kom puas tsuaj ntawm pathogens.
Yog hais tias ib koob tshuaj twb tsis tu ncua tshuaj tom ntej no koob tshuaj yog muab rau tog twg los coj sai li sai tau, ces ua raws li mounted regimen.
Sab los "Elefloks" tshuaj
"Levofloxacin" ( "Elefloks") tej zaum yuav ua txoj kev loj hlob ntawm sab los. Ntawm cov tau phiv tshua ntawm lub cev - lub tsos ntawm dysbiosis, tshuaj lom kab mob siab, enterocolitis, dyspepsia. Tej zaum yuav tam sim no nyob rau hauv cov leeg mob, mob plab, mob taub hau, raws plab, tu-sauv, tshee, kub. Thaum ib tug tsis zoo tshuaj tiv thaiv rau cov yeeb tshuaj nyob rau hauv lub siab enzymes, nce ua si yuav tsum muaj cai. Thaum nrhiav kom tau ntawm tej tshwm sim raws li pseudomembranous mob plab, ntxiv kev kho mob yuav tsis yooj yim sua.
Cov tshuaj no yog tej zaum nrog discoordination thaum ua taw, muaj cov kev xav lability, kev nyuaj siab, thiab pw tsaug zog teeb meem. Nyob rau hauv tej rooj plaub, pom teeb nco qab, cov kev txiav txim zoo ntawm tsis hnov tsw thiab saj. Mus rau daim ntawv teev kev phiv tshuaj muaj xws li arthralgia, thrombocytopenia. Tej zaum zoo tsim agranulocytosis, paresthesia. Tus neeg mob tej zaum yuav muaj leukopenia, eosinophilia.
Nrog kev xav txog lwm yam kev phiv thaum lub sij hawm kev kho mob "Elefloks" neeg saib xyuas muaj xws li cov lus qhia rau kev siv asthenic syndrome, hypoglycemia, kub taub hau, mob porphyria rau hauv cov duab, nce qab los noj mov, tachycardia, arrhythmia thiab ib tug tseem ceeb txo nyob rau hauv cov ntshav siab (muaj ib tug tau ntawm lub cev qhuav dej).
Tej zaum kuj muaj kev tsis haum tshuaj, muaj kub thiab khaus ntawm daim tawv nqaij, trembling ntawm lub nqua. Tau theem nrab kab mob. Nws yog ua tau lub tsos ntawm photosensitivity, neuropathy. Kom paub tias tej yam uas phiv - ib tug yog vim li cas rau kev kho mob rau cov kws kho mob.
Overdose "Elefloksa"
Txij li thaum muaj yog tsis muaj antidote, ib tug overdose ntawm symptomatic txoj kev kho yuav tsum tau. Ntawm cov zoo txoj kev mus rau tshem tawm xws li ib tug lub xeev - peritoneal kev lim ntshav, hemodialysis.
ceev faj
Cov neeg mob uas tseem tshuav tom qab kev kho mob txhais tau hais tias "Elefloks" tswv yim qhia ib tug faj siv ntawm cov tshuaj nyob rau hauv tej yam mob. Ib txhia neeg yuav tsum tau ib tug yuav tsum kho mob saib xyuas.
Nrog rau cov disappearance ntawm lub high school lub cev kub ntsuas txoj kev kho yuav tsum tau mus ntxiv rau lwm 2-3 hnub. Kev kho mob hnyav ncawv ntws mob ntsws yuav tsum tau siv li ntawm ob peb tshuaj, txwv tsis pub tus yam tshwm sim muaj peev xwm yuav rho.
Thaum lub sij hawm hauv chav kawm ntawm kev kho yuav tsum tsis txhob raug tus kab mob rau tshav ntuj thiab dag UV teeb vim hais tias ntawm txoj kev pheej hmoo ntawm photosensitivity.
Nws muaj lwm yam lus uas yuav tsum tau sai sai. Tej kev hloov rau kev kho mob yuav tsum qhia rau koj tus kws kho mob.
Lub ua ke ntawm "Elefloks" tshuaj nrog lwm yam tshuaj
Sib tham uas muaj tej yam tshuaj, "Elefloks" tej los yog thiaj li lawv cov nyhuv. Ib yam yuav tshwm sim rau cov kev txiav txim ntawm cov tshuaj. Yog hais tias tsim nyog, kev kho mob nrog rau lwm cov tshuaj nyob rau hauv cov kev kho mob lub sij hawm "Elefloksom" yuav tsum paub hais tias lawv tej zaum yuav tsis tau tshaj. Tej kev hloov txog cov tshuaj, yuav tsum tau tham nrog koj tus kws kho mob.
"Elefloksa" Nqi
Nyob ntawm seb ntau npaum daim ntawv "Elefloks" tshuaj nqi yog hais txog 760-940 rubles. rau cov ntsiav tshuaj nyob rau hauv ib tug ntau npaum ntawm 500 mg (№ 10). Hais txog 345-450 rubles. Nws yog tso dej tshuaj (100 mL).
Xyuas ntawm kev npaj "Elefloks"
Nyob rau hauv kev, cov neeg mob zoo soj ntsuam cov tshuaj. Raws li lawv, "Elefloks" yog npaum thiab ua rau nws tau los kho ntau yam kab mob ntawm cov kab etiology.
Cov tshuaj no feem ntau yog siv rau cov neeg mob mus tua nrog ob peb pathogens pathological tej yam kev mob yog tias tsim nyog.
Poob tom qab txoj kev kho txhais tau tias "Elefloks" cov lus teb qhia hais tias muaj cov uas tsis tshua muaj occurrences kev phiv tshuaj. Sab los feem ntau yog me me thiab ploj kiag li thaum txoj kev kho yog ua kom tiav.
Analogs "Elefloks" tshuaj
Tshuaj uas nws txiav txim yog zoo li ntawd muab rau lub cev "Elefloks", muaj nyob rau hauv loj naj npawb. Peb yuav paub qhov txawv cov tshuaj xws li "Maklevo", "Leobeg", "Lebel". Paub ntawm tau ntawm kev siv raws li ib tug kev hloov rau "Lefoktsina", "Levofloxacin", "Glewe", "Ivatsina". Cov nyiaj no yog cov feem ntau heev thiab yog siv los tos analogue rau cov tshuaj "Elefloks" yog hais tias tsim nyog. Nqe analogues hauv qab no, cov nyhuv ntawm lawv cov kev siv yog zoo sib xws.
"Elefloks" yog hais txog loj siv yeeb tshuaj thiab yuav ua ib tug ntau ntawm cov kev phiv. Ua ntej siv, nws yog ib qho tseem ceeb mus ua tib zoo nyeem cov lus qhia. Nws siv rau cov kev kho mob yuav tsum tau nqa tawm tsuas yog tom qab ib tug kws kho mob lub sij hawm teem tseg, uas yuav kom khiav ntawm cov kev hloov uas tshwm sim nyob rau hauv lub cev.
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