Noj qab haus huv, Npaj
"Vestikap": cov lus qhia rau kev siv. Drug analogues thiab kev xyuas txog nws
Cov lus qhia. Lub mechanism ntawm qhov kev txiav txim ntawm cov tshuaj
Txhais tau tias ntog mus rau hauv cov qeb ntawm histamine tshuaj. Lub active tshuaj influences lub H3 thiab H1-receptors nyob rau hauv lub Cns thiab vestibular nuclei nyob rau hauv lub inner pob ntseg. Los ntawm ncaj qha agonistic txiav txim, paub permeability thiab microcirculation nyob rau hauv cov hlab ntsha, stabilized nyob rau hauv lub cochlea thiab labyrinth siab endolymph. Nyob rau tib lub sij hawm muaj ib qho kev nce ntawm cov ntshav khiav tsis zoo hauv lub basilar leeg. Tshuaj accelerates rov qab los ntawm kev ua tom qab unilateral vestibular neyrektomii. Cov nyhuv no yog vim kev thaiv kev nrog histamine H3 receptor. Qhov no tswj thiab accelerates lub hauv paus vestibular nyiaj. Lub medicament "Vestikap" (phau ntawv qhia no muaj cov ntaub ntawv xws li) muaj ib tug hais central nyhuv, koob tshuaj-dependent decreases nyob rau hauv neurons ntawm lub nrub nrab thiab lateral vestibular nuclei tiam tej zaum. Cas kho nyhuv yog cai tom qab ob lub lis piam.
pharmacokinetic zog
Txhais tau tias undergoes sai haum. Muaj tsawg daim ntawv cog lus nrog ntshav proteins. Tsis pub dhau peb teev lub concentration ntawm cov tshuaj nyob rau hauv cov ntshav nce mus txog ib tug tshaj plaws. Nyob rau hauv tus txheej txheem ntawm lwj ua 2-pyridylacetic acid thiab demetilbetagistin. Yuav luag tag (80-90%) tas los ntawm ob lub raum thaum lub sij hawm ib hnub. Ib tug me ib feem ntawm cov hniav lwj cov khoom tso tawm kom pom los ntawm cov hnyuv.
lub sij hawm
Tshuaj "Vestikap" phau ntawv qhia xav kom Meniere lub syndrome, nrog los ntawm tinnitus, tsis hnov lus thiab kiv taub hau. Cov tshuaj zoo eliminates xws ces complicating mob, raws li xeev siab thiab retching. Tshuaj qhia rau cov symptomatic kev kho mob ntawm Kiv tauv hau (kiv taub hau ntawm vestibular keeb kwm).
Contraindications
Nws txhais tau hais tias tsis pom zoo thaum glucose intolerance, npau taws me ntsis rau Cheebtsam txhais tau tias lactation. Kev kho mob yog contraindicated rau cov poj niam xeeb tub, mis-pub mis. Tsis prescribers "Vestikap" (phau ntawv qhia ceeb toom txog nws) nyob rau hauv thaum yau. Pub cov neeg mob yuav tsum tau rau lub caij ntawm txoj kev kho kom tsis txhob pub. Ceev faj thaum lub sij hawm txais tos yuav tsum muaj cai nyob rau hauv lub xub ntiag ntawm ulcerative txhab ntawm lub digestive system (keeb kwm xws li), bronchial hawb pob, feohromtsitome. Cov neeg mob nrog cov saum toj no pathologies yuav tsum tau kho nyob rau hauv ze kho mob saib xyuas. Nyob rau hauv tej rooj plaub, tej zaum nws yuav yuav tsum tau kev kho me ntsis nyob rau hauv ntau npaum regimen.
dosing regimen
Medicament "Vestikap" phau ntawv qhia xav haus thaum lub sij hawm noj mov. 8 mg tsiav tshuaj nyob rau hauv ib tug-lub sij hawm ntau npaum ntawm 2.1 units nyob rau hauv 16 mg -. By 1 piece. Txhais tau hais tias noj peb zaug ib hnub twg. Feem ntau, cov kev txhim kho los ntawm thaum ntxov ua sawv ntawm txoj kev kho. Txawm li cas los, ib tug ruaj khov nyhuv cai tom qab kaum plaub hnub. Rau ob peb lub hlis, cov tshuaj yuav muaj kev nce. Duration ntawm kev kho mob. Duration ntawm lub Hoob no yog teem ib lub zuj zus tshwj xeeb.
phiv
Cov tshuaj provokes mob plab, ntuav, angioedema (muaj tsawg heev). Cov nyom zoo xws li dyspepsia, flatulence, tawm pob. Nyob rau hauv cov ntaub ntawv ntawm cov kev phiv tshuaj yuav tsum tau nrog ib tug tshwj xeeb. Thaum pom tau hais tias cov tshuaj overdose ntxias cov exacerbation ntawm cov tsos mob. Qaug cawv yog nrog los ntawm tsaug zog (nyob rau hauv cov ntaub ntawv uas tau txais mus rau 640 mg ntawm yeeb tshuaj), kab mob (thaum noj ntau tshaj 640 mg los sis nyob rau hauv ua ke nrog nrog rau lwm cov medicaments). Nyob rau hauv xws li mob, symptomatic kev kho mob yog taw, thiab qhov yuav tsum tau mus xyuas ib tug kws kho mob. Nrog raws sij hawm kev kho mob cov kws ho thiaj li qhov uas yuav muaj teeb meem thiab cov tsos mob ntawm intoxication yog tshem tawm nyob rau hauv ib tug luv luv lub sij hawm. Raws li ib tug thawj pab ntsuas pom zoo pais plab lavage.
Yuav ua li cas yuav hloov tau cov tshuaj? Cov feem nrov analogues
"Vestikap" - raws li histamine tshuaj series - muaj ib tug ntau ntawm tshuaj-txhais (los yog generic), muaj ib tug zoo kho nyhuv. Qhov zoo tshaj plaws kev xaiv yuav kho tau tus thawj txhais tau tias "Betaserk". Txawm li cas los, nyob rau hauv kev sib piv nrog rau lwm cov tshuaj no yog kim heev (txog 400-600 rubles). Cov feem nrov thiab pheej yig tshuaj nyob rau hauv Russia, uas yuav tsum tau hloov los ntawm txoj kev "Vestikap" yuav tsum muaj xws li tshuaj "Tagista" thiab "Vestibo". Lawv tag nrho cov muaj ib tug active tshuaj, albeit nyob rau hauv sib txawv ntau. Nyob ntawm seb nws cov ntsiab lus, thiab tus nqi yog muab.
Tshuaj "Vestibo"
Muaj nyob rau hauv cov ntsiav tshuaj daim ntawv. Cov tshuaj muaj ib tug me me agonistic ntxim rau H1 receptors. Medicament exhibits vasodilatory thiab gistaminpodobnuyu kev ua si. Hais tias ib tug heev haib ntxim rau cov H3 receptors. Cov tshuaj tsis ua koj nkees nkees thiab sedative los, raws li ib co lwm yam analogues "Vestikap". Txhais tau hais tias "Vestibo" yog tsis pom zoo thaum lub sij hawm thawj peb lub hlis, nrog ceev faj (rau kev kho mob yog vim li cas), taw thaum lub sij hawm thib ob thiab thib peb trimesters ntawm cev xeeb tub.
"Tagista" tshuaj
Lub medicament yuav muab ob qho tib si raws li ib tug kev kho mob thiab kev tiv thaiv ntawm vestibular kiv taub hau txawv etiology. Cov tshuaj no kuj muaj nyob rau hauv cov ntsiav tshuaj daim ntawv. Contraindications muaj xws li cov hnub nyoog ntawm 18 xyoo, cev xeeb tub. Tsis txhob muab tshuaj lactating cov neeg mob. Thaum tau txais txhais tau tias tej zaum yuav muaj ib tug teeb meem ntawm tus mob huam ua si, npau taws me ntsis kev tshua, angioedema.
Yuav ua li cas hais txog cov "Vestikap 'tshuaj xyuas?
Nyob rau hauv kev, nrog rau kev hwm mus tolerability ntawm cov tshuaj, cov lus ntawm cov neeg mob qhia tias lub chaw tshua ntxias phiv. Sawv pliaj los yuav muab tshem tawm tom qab lub abolition ntawm cov tshuaj thiab tsis yuav tsum tau ntxiv kev pab. Nyob rau hauv cov ntaub ntawv no, cov kws txawj hais tias
Yog xav paub ntxiv,
Medicament "Vestikap" haum rau kev siv rau peb lub xyoos. Khaws cov tshuaj yuav tsum tau nyob rau hauv ib tug maub qhov chaw, deb ntawm cov me nyuam. Kub yuav tsum tsis txhob yuav ntau dua 25 degrees. Kws txawj nco ntsoov tias cov tshuaj "Vestikap" raws li zoo xws li cov tshuaj ntawm no pab pawg neeg yog suav tias yog muaj zog txaus yeeb tshuaj, txawm lub fact tias nyob rau hauv tej rooj plaub tsim maj. Txhais tau hais tias ua ib tug "Nws" Lavxias teb sab kws lub tuam txhab. Tus nqi ntawm cov tshuaj mas nws txawv nyob rau hauv ntau ntawm 150 rau 200 rubles (los yog ntau tshaj). Txhais tau hais tias cov tshuaj.
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