Noj qab haus huvNpaj

"Itraconazole": kev qhia, pheej yig analogues, txheeb xyuas thiab kev tso tawm daim ntawv no. Analog "itraconazole" ntsiav tshuaj. "Itraconazole" (tshuaj pleev): counterparts

Kev npaj "Itraconazole" (ntsiav tshuaj, tshuaj pleev, cream, tov los tsiav tshuaj) yog siv rau cov kev kho mob los ntawm ntau yam fungal kab mob. Nyob rau tib lub sij hawm nws yog Attendance zoo rau cov kev kho mob ntawm cov kab mob uas yog laus nyob rau hauv ntau qhov chaw ntawm lub cev.

Cov tshuaj tshuaj

Kev npaj nws tus kheej thiab tej analogue "Itrakanozola" yog hais txog ib tug hauv chav kawm ntawv ntawm noj triazoles. Qhov no artificially tsim tshuaj tiv thaiv lub synthesis ntawm ergosterol yuav tsum tau rau qub hauj lwm ntawm fungi. Tshuaj "Itraconazole" suppresses txoj kev loj hlob dermagofitov, yeasts ntawm Candida, fungi thiab lwm yam pathogens. Ib txhia kab mob los ntawm kab mob resistant rau no neeg sawv cev.

Kev npaj "Itraconazole" yog muaj nyob rau hauv cov ntsiav tshuaj, tsiav tshuaj, raws li ib tug tshuaj (kua) tshuaj pleev. Kev muag khoom yog nyob deb ntau tshaj ib tug analogue "itraconazole". Zoo li npaj yog muaj nyob rau hauv ntau yam ntau npaum cov ntaub ntawv.

Tej analogue "itraconazole" thiab, nyob rau hauv qhov tseeb, cov kev npaj nws tus kheej yog feem ntau siv rau cov kev kho mob ntawm fungal kab mob ntawm lub pa system, tshwj xeeb tshaj yog lub ntsws. Cov tshuaj no siv tau rau cov kev kho mob ntawm cov neeg uas ntaus fungi caj pas, qhov ncauj kab noj hniav los yog txoj hlab nqos mov. Heev feem ntau, tus kab mob no muaj feem xyuam rau cov tib neeg tes. Nyob rau hauv cov ntaub ntawv no, siv ib tug txawv ntau npaum daim ntawv "Itraconazole" tshuaj - ib tug tshuaj pleev rau lwm siv, uas zoo, khoom fungal kab mob ntawm lub tes los yog daim tawv nqaij. Nws muab thiab psoriasis.

indications

Qhov no siv yeeb tshuaj thiab nws analogues yog siv nyob rau hauv cov nram no cov kab mob:

• mob txhab txiag;

• Candidiasis;

• sporotrichosis;

• pityriasis versicolor;

• onychomycosis;

• blastomycosis;

• cryptococcosis;

• keratomikoz;

• paracoccidioidomycosis;

• mauj aspergillosis thiab Candidiasis;

• histoplasmosis;

• tauj mycoses.

Lub caij ntawm txoj kev kho tej zaum yuav tau tom nyob ntawm tus soj ntsuam daim duab. Feem ntau cov feem ntau, cov tshuaj no yuav tsum tau coj ib lub sij hawm ib hnub twg. Cov feem ntau siv kev kho mob kiag:

• chromophytosis: thaum lub sij hawm lub lim tiam, 200 mg;

• mob txhab txiag: thaum lub sij hawm lub lim tiam, 200 mg los yog 100 mg rau 15 hnub;

• onychomycosis 3 lub hlis ntawm 200 mg txhua lub limtiam los yog 200 mg / 2 lub sij hawm ib hnub twg;

• Tinea ntawm ob txhais tes thiab ob txhais taw: ib lub lim tiam ntawm 200 mg los yog 100 mg rau 1 lub hli;

• Candidiasis: 15 hnub, 100 mg;

• keratomikoz: 3 lub lim piam ntawm 200 mg.

Txoj kev rau txais tos nyob rau hauv pulmonary kab mob

Rau cov kev kho mob ntawm fungal kab mob "Itraconazole" caj pas muab ntsiav tshuaj los sis tsiav tshuaj. Analogs yog pheej yig dua, tab sis tej zaum lawv yuav muaj ib tug ntau nyob deb nyob rau hauv lub sij hawm qhov kev txiav txim, ces tus kab mob no yog yam nyuab dua los yeej sai li sai tau. Ntsiav tshuaj los yog tshuaj noj 1-2 lub sij hawm ib hnub twg, thaum lub sij hawm los yog sai li sai tau tom qab ib tug noj mov. Feem ntau, rau cov kev kho mob ntawm fungal kab mob ntawm lub ntsws yuav tsum tau ib tug tsawg kawg nkaus ntawm 3 lub hlis. Nyob rau hauv tej rooj plaub, tus kws kho mob yuav muab tshuaj rau tom ntej no chav kawm ntawm kev kho mob: 3 ntsiav tshuaj ib hnub twg rau 3 hnub, ua raws li los ntawm 3 lub hlis ntawm 1-2 ntsiav tshuaj ib hnub twg.

Noj cov tshuaj nrog tus ntsia thawv kab mob

Tshuaj "Itraconazole" - tshuaj uas yog kws kho rau cov kev kho mob ntawm fungal ntsia thawv kab mob. Rau ib tug tag nrho kev kho nws yog coj 1 lub sij hawm ib hnub twg rau 12 lub lis piam. Ntau zoo yog lub qhov ncauj tov "Itraconazole". Nws yog muab rau 1-4 lub lis piam, 1-2 zaug ib hnub twg. Nyob rau hauv tas li ntawd, rau ib tug ntau ceev ceev haum ntawm cov tshuaj noj rau ib qho kev npliag plab. Xaiv lub feem ntau pom dosing tswvyim los yog xaiv analogue "itraconazole" tsuas yog muaj peev xwm sawv ntawm tus kws kho mob, uas yuav coj mus rau hauv tus account nyob rau hauv cov ntaub ntawv no heev ntawm tus kab mob thiab lub xeev ntawm tus neeg mob. Nyob rau hauv lub feem ntau loj heev zaum los kho fungal kab mob ntawm lub tes siv lwm daim ntawv ntawm "Itraconazole" tshuaj - ib tug tshuaj pleev uas yog thov mus rau lub cheeb tsam cov 1-2 zaug ib hnub twg.

Lwm yam embodiments ntawm cov tshuaj

Tej analogue "itraconazole" nws tus kheej ntawm cov tshuaj no nyob rau hauv xyoo tsis ntev los nce siv nyob rau hauv cov kev kho mob ntawm ntau hom ntawm fungal kab mob nyob rau hauv cov neeg mob cuam tshuam los ntawm tus kab mob HIV thiab AIDS. Nyob rau hauv cov ntaub ntawv no tsis tsim nyog nws tus kheej, vim hais tias tsuas yog tus kws kho mob yuav kom ntsuam xyuas tus neeg mob lub noj qab haus huv thiab tau uas tau txais "itraconazole" txaus ntshai.

ceev faj

Tshuaj "Itraconazole" analogues cov tshuaj no yuav tsum tau noj nyob rau hauv raws li cov lus qhia thiab cov tswv yim ntawm cov kws kho mob. Nyob rau hauv me me los yog loj koob tshuaj tej zaum yuav pab tsis tau los yog muaj peev xwm ua mob rau tus neeg mob lub cev.

Tsiav tshuaj "Itraconazole" analogues ntawm pheej yig los yog kim yog npaum li cas raws li nram no: tsiav tshuaj thiab cov ntsiav tshuaj yog nqos tag nrho. Nyob rau tib lub sij hawm lawv yuav tsum tsis txhob zom lossis zuaj. Los ntawm kev txo qhov theem ntawm acidity nyob rau hauv lub plab, tshwm sim los ntawm, piv txwv li, cystic fibrosis, yuav tsum tau qhia rau koj tus kws kho mob.

Nyob rau hauv tej rooj plaub, lub regimen ntawm cov tshuaj yuav tsum tau muab hloov. Feem ntau cov feem ntau qhov no tshwm sim thaum twg, thaum lub sij hawm txoj kev kho tus neeg mob yog noj cov nram qab no tshuaj: "famotidine", "nizatidine", "esomeprazole", "cimetidine", "omeprazole", "Ranitidine", "Lansoprazole", "pantoprazole", " rabeprazole. "

Contraindications

Nyob rau hauv tej rooj plaub, cov neeg mob yuav txhob "Itraconazole". Coj zoo xws li cov tshuaj feem ntau txwv tsis pub xws noj tshuaj rau tsis haum lawv lub Cheebtsam. Uas yog vim li cas lub sij hawm ntawm txoj kev kho nrog cov tshuaj tus kws kho mob yuav tsum paub raws nraim seb ib tug neeg mob muaj yog ib tug tsis haum cov tshuaj tiv thaiv rau ib yam khoom uas muaj nyob rau hauv lawv cov muaj pes tsawg leeg.

Tshuaj yuav tsum tsis txhob yuav npaum li cas los cev xeeb tub los yog lactating cov poj niam. Yuav kom tiv thaiv tau ib tug tau cev xeeb tub thaum lub sij hawm kev kho mob yog tsim nyog los siv txhais tau tias zoo ntawm pov. Nrog kev saib xyuas active tshuaj los siv rau cov neeg laus cov neeg mob. Tau txais nws thaum yau yog tau tsuas yog thaum cov kev pab ntau tshaj tej zaum yuav raug. Cov tshuaj no yog tsis pom zoo rau cov neeg mob plawv tsis ua hauj lwm, ischemia, mob ntsws kab mob, lub raum insufficiency.

"Itraconazole" analogues ntawm cov tshuaj yuav tsum tsis txhob coj nyob rau hauv ib tug muab ob npaug rau koob tshuaj, nrog rau cov tau tso cai ntawm lub tshuaj. Nws yog qhov zoo tshaj plaws tsis nco txog kev tsis koob tshuaj thiab ua raws li cov regimen. Peb yuav tsis cia ib tug overdose ntawm cov tshuaj, los yog nws analogues, raws li qhov no yuav ua tau kom mob loj heev noj qab haus huv mob.

Sis nrog lwm yam tshuaj

Ua ntej yuav noj "itraconazole" tus kws kho mob yuav tsum tau paub txog dab tsi tshuaj tus neeg mob noj ua ntej. Tshwj xeeb tshaj yog nws kev txhawj xeeb rau kev siv ntawm tej cov tshuaj raws li "Efavirenz", "Everolimus", "sildenafil", "Aliskiren", "Rifabutin", "apixaban", "NVP", "Dasatinib", "Ibrutinib", "Salmeterol", " darifenacin, "" Nilotinib "," Karbazepin "," Sunitinib "," Colchicine "," Rivaroxaban "," Phenobarbital "" Tamsulosin "," Isoniazid "," Phenytoin "" Vardenafil "," Rifampicin "," NVP " "Temsirolimus".

Nyob rau hauv tas li ntawd mus rau cov khoom ua ntej yuav siv "itraconazole" yuav tsum qhia rau koj tus kws kho mob txog kev noj cov nram qab no:

• anticoagulants;

• tshuaj tua kab mob;

• HIV protease inhibitors;

• vitamins;

• noj tshuaj pab (noj tshuaj pab).

Nrog simultaneous siv "itraconazole" thiab antacids yog siv rau lub 1 teev ua ntej los yog tom qab ib tug ob peb teev tom qab thawj coj ntawm noj tshuaj.

phiv

Tshuaj "Itraconazole" tej zaum yuav ua rau kiv taub hau thiab qhov muag plooj tsis pom kev nyob rau hauv daim ntawv ntawm ib tug split duab. Thaum tau txais cov tshuaj yuav tsis tsav ib lub tsheb, thiab ua hauj lwm nrog ntau cov khoom siv. Cov feem ntau qhia phiv txheej xwm thaum noj muaj xws li tsam plab, flatulence, raws plab, quav tawv, kub siab, tshwm sim los ntawm ib tug unpleasant saj nyob rau hauv lub qhov ncauj; nce tawm hws, kiv taub hau, mob taub hau, los ntshav thiab mob cov pos hniav, mob nyob rau hauv cov nqaij, poob nqaij laus, los ntswg qhov ntswg, ua npaws, mob tej pob txha, kev nyuaj siab, poob libido, tsis ntawm cov plaub hau.

Tshwj xeeb yog txaus ntshai rau cov kev kho mob ntawm tus neeg mob yog cov nram no phiv: muab ob npaug rau pom kev, hnov xeev xeev siab, ntuav, tu-sauv nyob rau hauv lub plab mog, lub plawv tsis ua hauj lwm, kab mob siab, mob txeeb tuskheej, anaphylactic thiab kev tsis haum tshuaj, tso zis dub, ringing nyob rau hauv lub pob ntseg, tsis hnov lus, tsis qab los noj mov, ntev li qaug zog , daj ntawm daim tawv nqaij thiab ob lub qhov muag, xws li loog loog thiab tingling ntawm daim tawv nqaij thiab nqaij mos mos, photophobia, daim tawv nqaij ua pob liab vog, khaus, txhaws qa, pulmonary edema, coj khaub mob, o ntawm lub ntsej muag, caj pas, ob txhais tes, pob taw. Yog hais tias koj muaj tej yam ntawm lub saum toj no cov tsos mob, qhov no yuav tsum tau qhia sai li sai tau rau koj tus kws khomob.

Yuav ua li cas los xaiv ib tug analogue "itraconazole"

Txhua txhua xyoo ntau thiab ntau cov neeg muaj txojkev qhov teeb meem ntawm fungal kab mob. Txawm li cas los, muaj ntau yam cov neeg mob txiav txim siab yog dab tsi los kho rau lawv tsis tas tau "Itraconazole". Analogs pheej yig dua, yog li ntawd lawv feem ntau dua. Nyob rau hauv qhov tseeb, cov lus nug ntawm kev xaiv ntawm cov tshuaj yeeb los yog nws analogues yuav tsum tau txiav txim siab xwb los ntawm lub mus kawm tus kws kho mob. Nyob rau hauv ib co loj heev zaum, tus neeg mob lub tag nrho rov qab yuav pab tau heev "Itraconazole". Analogs ntawm pheej yig, tab sis tsis yog txhua txhua ntawm lawv yog cov zoo li raws li cov tshuaj.

Ib yam yuav tsum tau hloov los ntawm "Itraconazole"? Tshuaj pleev, analogs ntawm lub cuab tam nyob rau hauv lwm yam ntau npaum ntawv no muaj nyob rau hauv khw muag tshuaj. Cov yam ntxwv analogs muaj xws li tshuaj manufactured nyob rau hauv lub pub tsiav tshuaj "Irunine", "Intramikol", "Itrazol", "Mikonihol", "Kanditral", "Kanazol", "Teknazol", "Orungal", "Rumikoz", "Orungamin "," Orun ".

Analogs "itraconazole" rau kho txiav txim yog cov nram no cov khoom:

  • Tsiav tshuaj "Diflucan", "Diflazon", "Itrazol", "Orungal", "Rumikoz", "Flucostat" "Fluconazole", "Fungolon";
  • ntsiav tshuaj "Atifin", "Binafin", "Ketoconazole", "Fungoterbin", "Ekzifin", "Nizoral";
  • tshuaj pleev, cream, tshuaj kua, "Akriderm" "Lamisil Dermagel", "Terbizil", "Ekzifin", "mikomaks", "Mikozoral", "Triderm", "Fungoterbin", "Ketoconazole", "Canison", "Lamitel" "candid", "Amiklon", "Zalain", "Canison", "Atifin", "Clotrimazole" "Lamisil" "Ifenek", "Lamitel", "Terbiks", "imide";
  • suppositories, paum ntsiav tshuaj, "Zalain", "Candide", "Canison", "Mikogal", "imide".

Xyuas

Yuav ua li cas yog koj lub tswv yim nyob rau hauv cov neeg noj cov tshuaj "Itraconazole"? Analogues, uas xyuas yog feem ntau ib tug tsis zoo connotation, thiab qhov chaw uas cov tshuaj no feem ntau tsis coj cov kev tsim tau los ntawm txoj kev kho. Nyob rau hauv cov ntaub ntawv no, tus loj tus naj npawb ntawm contraindications thiab kev phiv ua cov tshuaj yog heev txaus ntshai rau lub noj qab haus huv ntawm ntau cov neeg mob. Ntxiv mus, txoj kev pheej hmoo ntawm tsis kaj siab txim ntawm txoj kev siv ntawm "itraconazole" thiab nws cov analogues yog ho muaj zog uas tsis yog raws kev cai nrog cov lus qhia ntawm tus kws kho mob los yog nws tus kheej-medicate.

Heev feem ntau muaj cov tsis zoo xyuas txog cov tshuaj "Itraconazole" (taws tswm ciab). Analogs ntawm cov tshuaj no feem ntau kuj ntaus nqi los ntawm cov neeg mob uas ceev faj. Qhov no yog vim lub fact tias nyob rau hauv tej rooj plaub cov kev kho mob ntawm fungal kab mob nrog rau cov kev pab los ntawm tswm ciab yuav tsum tau complemented los ntawm kev noj "itraconazole" los yog analogs hauv.

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