Noj qab haus huv, Npaj
Analogs "Atoris": hauj lwm, xyuas
Tshuaj "Atoris" sau npe ua khoom ntawm lub Slovenian kws lub tuam txhab "KRKA". Nws yog ib tug zoo thiab pheej yig generic "atorvastatin", uas yav tas los tsuas muag raws li ib tug tshuaj ntawm Pfizer 'Lipitor'. Thaum lub caij, nws analogs ( "Atoris", "Torvakard" thiab lwm tus neeg) tau ua ib feem ntawm kev soj ntsuam xyaum thiab zoo yog hypocholesterolemic agents.
muab
Kev npaj "Atoris" yog muaj nyob rau hauv cov ntsiav tshuaj ntawm peb tsev noj tshuaj npaum cas. Qhov no 10, 20 thiab 40 mg. Muag nyob rau hauv cartons, nrog kev pab nyob rau hauv sawv hlwv ntsiav tshuaj. Peev Xwm ntawm cartons 10, 30 thiab 90 'Atoris "ntsiav tshuaj (phau ntawv qhia). Analogs generic tshuaj thiab tej zaum yuav muaj tib yam nqi ntawm active tshuaj, tiam sis tsis muaj cov nyhuv tib vim yog txawv nyob rau hauv lub Cheebtsam.
Cov tshuaj "Atoris"
Lub active tshuaj yog atorvastatin, statin III tiam. Koom haum pab tshuaj yog cov nram qab no: polyvinyl cawv, titanium dioxide, macrogol 3000, magnesium stearate, talc, croscarmellose sodium, microcrystalline cellulose, lactose monohydrate, povidone, calcium carbonate, sodium lauryl sulfate.
Cam txiav txim tableted ntau npaum daim ntawv thiab txiav txim seb tus nqi ntawm atorvastatin haum mus rau hauv cov hlab ntsha. Raws li, tej analog tshuaj "Atoris" yuav tsum muaj tus nqi qub active tshuaj tso tawm thiab nyob rau tib lub ceev, tsim zoo xws li cov ntshav ntau.
Ua neeg ncajncees ntawm statins thiab tshuaj "Atoris"
Kev npaj "Atoris" raws li active tshuaj muaj atorvastatin. Nws belongs rau hauv qeb ntawm peb-tiam agents. Nrog nws nyob ntau ntau ntawm cov kev tshawb fawb uas tau paub tseeb hais tias cov feasibility ntawm nws txais tos nyob rau hauv lub xub ntiag ntawm atherosclerosis muaj tej yam los sis twb tsim tus kab mob no. "Atorvastatin" analogs, "Atoris" thiab lwm yam statins txo lub peev xwm ntawm cov uas tsis muaj kev ceev lipoproteins (LDL) ua rau atherosclerosis thiab ua rau nws cov aggravation. Qhov no yog lawv cov kev soj ntsuam nqi, vim hais tias nrog lawv mus koom tes thiaj li cov xwm txheej ntawm cov lub plawv tuaj.
pharmacological los
Qhov tseem ceeb tshaj qhov yuav tau txais ntawm tau txais ib tug muaj kev nyuaj siab ntawm cholesterol synthesis los ntawm inhibiting lub enzyme HMG-CoA reductase. Cov no ib tug txiav los tseem ceeb yuav txo tau nyob rau hauv lub synthesis ntawm LDL. Qhov no feem ntawm lipoproteins ntxias atherosclerosis, ua narrowing ntawm cov phab ntsa thiab nws cov kev foob nyob rau hauv cov hlab ntsha ntawm lub plawv, lub hlwb thiab sab nqua. Ua ke nrog cov yuav txo tau ntawm LDL tsub kom lub concentration ntawm kev kub ceev lipoproteins.
Lawv ua hauj lwm tseem ceeb: nce membrane kuj mus txhua yam thiab tshuaj influences vim lub incorporation ntawm cholesterol mus rau hauv nws. Yog li, HDL pov tseg, tab sis tsis ntxiv roj uas txhaws taus. LDL ua rau nws cia hnab khib qab lub vascular endothelium, ua arteriosclerosis, thaum high-density lipoprotein cholesterol deposits txo tus nqi, tab sis ua tsis tau tso zis nws ntawm lub puab plhaub leeg elastic hom.
Dosing "Atoris" npaj
Pom zoo nyob rau hauv yuav ua li cas coj "Atoris" rhaub cia hais tej yam. Nyob rau hauv kev, cov tshuaj yog coj nyob rau hauv lub kws tshuaj ib hnub ib zaug tom qab noj hmo ua ntej yuav mus pw. Ib tug tib koob tshuaj yuav ua tau 10, 20 thiab 40 mg. Txij li thaum cov tshuaj yog ib cov tshuaj rau nws purchase yuav tsum tau sab laj ib tug kws kho mob. Hais tias nws tom qab tsom xam thiab kev ntsuam xyuas ntawm lipid profile zauv feem ntawm tag nrho cov ntshav cholesterol theem yog tau pom zoo kom tau qhov tseeb ntau npaum ntawm atorvastatin thiab nws analogs los yog generic chav kawm ntawv.
Thaum thawj zaug cholesterol theem ntawm 7.5 los yog ntau dua yog pom zoo kom noj 80 mg / hnub. Zoo li ntau npaum tus kws kho rau cov neeg mob uas tau raug kev txom nyem ib myocardial infarction los yog nyob rau hauv lub mob nyob ntev ntawm nws cov hoob kawm. Thaum ib tug concentration ntawm 6.5 rau 7.5 pom zoo koob tshuaj yog 40 mg. 20 mg thaum lub cholesterol theem ntawm 5.5 - 6.5 mmol / liter. 10 mg ntawm cov tshuaj haum rau cov me nyuam los ntawm 10 mus rau 17 xyoo uas muaj heterozygous hypercholesterolemia, raws li zoo raws li cov laus uas thawj hypercholesterolemia.
Yuav tsum muaj rau Generics
Zoo analogue "Atoris" kev npaj yuav muaj ib qho zoo tib yam kom muaj nuj nqis ntawm active ingredient thiab tsim zoo xws li cov ntshav ntau. Yog tias cov txhais tau tias yog zoo li no, nws yog tswv kom yuav bioequivalent thiab yuav hloov cov thawj kiag li. Nrog kev hwm rau cov tshuaj "Lipitor" yog ib tug analogue ntawm "Atoris", tsim nyob rau hauv lub hauv paus ntawm atorvastatin.
Yuav tsum muaj rau kev soj ntsuam analogues "Atoris"
Tej kev hloov "Atoris", nws chav kawm ntawv los yog sib npaug nyob rau hauv muaj pes tsawg leeg, yuav tsum muaj ib yam ntawm cov statins. Nyob rau hauv cov ntaub ntawv no, nws yuav siv tau raws li ib tug tag nrho cov sib npaug. Ntxiv mus, cov kev hloov ntawm "Atoris" tshuaj rau lub analogue yuav tsum tau nqa tawm nrog lub npaj ntau npaum ntawm preservation. Yog hais tias koj siv 10 mg "Atoris", ces lwm cov tshuaj yuav tsum tau ua tib yam los yog ntau dua ua si.
Generic "Lipitor"
Txij li thaum tus thawj atorvastatin yog "Lipitor" tag nrho cov tshuaj uas muaj tib lub active ingredient yuav tsum tsis txhob piv nrog nws. Analogs, "Atoris" cov uas lub feem ntau balanced nyob rau hauv tus nqi, yuav tsum tau raug xam tias yog los ntawm qhov no taw tes ntawm view. Yog li ntawd, muaj xws li medicaments dua tus nqi, nrog ib tug sib npaug thiab ib tug tsawg dua. Tag nrho cov analogues "Atoris":
- kim ( "Lipitor");
- Attendance mus siv cuag ( "Torvakard", "Tulip");
- cheaper ( "Lipromak", "Atomaks", "Lipoford", "Liptonorm").
Raws li yuav pom, atorvastatin analogues lug sawv cev. Muaj ntau ntau yog muaj nyob rau hauv cov uas tsis muaj nqi qeb. Qhov no yuav tsum muaj xws li ib tug ntau ntawm cov tshuaj nrog cov lag luam tawm npe "Atorvastatin", uas yog ua nyob rau hauv daim ntawv tso cai los ntawm loj kws tuam txhab uas muag.
Yog hais tias peb nrhiav kom tau ib tug analogue ntawm "Atoris" cheaper atorvastatin yog tej domestic ntau lawm nyob rau hauv daim ntawv tso cai. Qhov tseem high-zoo thiab tag nrho raws li cov kev piav yog "Atorvastatin" Borisov cog ntawm pharmaceuticals, yog nyob rau hauv Belarus. Ntawm no, zus tau tej cov tshuaj yog tshuaj los ntawm KRKA, uas ua "Atoris".
Nta ntawm cov kev hloov cov tshuaj
Nyob rau cov nqe lus nug ntawm yog dab tsi los hloov "Atoris", nws yog ib qho tseem ceeb uas yuav tau xav ob peb yam kev mob. Thawj, cov tshuaj yuav tsum tau muaj ib tug haum soj ntsuam miv nyuas siv zug thiab zoo taus. Secondly, nws cov nqi yuav tsum yog tsawg dua, los yog hais tias cov tshuaj hauv chav kawm ntawv koom rau analogs me ntsis saum toj no. Thirdly, lub yav tas koob tshuaj yuav tsum tau ua raws li, yog tias ib tug hloov yog ua rau cov generic. Nyob rau hauv cov ntaub ntawv ntawm qhov kev hloov rau ib tug analogue ntawm cov tshuaj hauv chav kawm ntawv nws yog ib qho tseem ceeb kom tau ib npaug koob tshuaj.
Hloov rau Generics
Cov kev npaj uas muaj atorvastatin, yog cov feem ntau zoo li nram qab no: "Lipitor" "Torvakard", "Lipromak" thiab "Atoris". Analogs, xyuas uas yog scarce, ua tsis tau zoo rau lawv nyob rau hauv miv nyuas siv zug thiab kev nyab xeeb. Txawm tias lawv yog cov nqi nyiam. Lawv yuav tsum tau pom zoo rau cov neeg mob uas tsis care txog lub bioequivalence ntawm generic los yog tsis xav kom overpay. Pom sib txawv nyob rau hauv cov nyhuv ntawm no yog tsis pom, txawm hais tias tus zoo ntawm kev kho mob rau ib co raws li cuam tshuam.
Yog hais tias peb xav txog cov generic atorvastatin, nws yog pom zoo kom xaiv los ntawm cov saum toj no. Tab sis, piv txwv li, los mus txiav txim seb yuav ua li xaiv - yog tsis yooj yim, "Atoris" los yog "Torvakard". Yog vim li cas rau qhov no yog qhov yuav luag tiav raws li cov tshuaj nyob rau hauv nqe thiab zoo heev. Ntxiv mus, tus nqi yog feem ntau kuj zoo sib xws. Saum toj no lawv yog qhov zoo tshaj ntawm "Lipitor" thiab hauv qab no - "Lipromak". Nyob rau tib lub sij hawm kawg, nrog ib tug me ntsis txawv nyob rau hauv cov khoom xyaw, pheej yig dua.
Hloov chav kawm ntawv counterparts "Atoris"
Nyob rau hauv kev npaj "Atoris" analogues nyob rau hauv Ukraine thiab lwm yam CIS lub teb chaws, tseem muaj cov hoob kawm. Uas yog, cov kev npaj muaj lwm statin, ntsig txog, uas txawv yam ntxwv. Qhov tseem tsim nyog hloov "Atoris" mus rau "pitavastatin" los yog "Rosuvastatin" nrog ib tug me ntsis degree ntawm LDL txos. Cov yav tas yog kev ruaj ntseg thiab muaj ib tug kho nyhuv ntawm ib qis koob tshuaj.
ua ntej lawm counterparts, tseem muaj "Atoris" yog ntau preferable nyob rau hauv kev sib piv nrog lawv, txawm hais tias lawv muaj ib tug soj ntsuam cov nyhuv rau lub hom phiaj zoo. Piv txwv li, "Simvastatin" - lub feem ntau pheej yig tshuaj nrog pov thawj raug soj ntsuam kev ruaj ntseg. Tus thawj qhov chaw yog 'Zocor'. Yog hais tias peb xav txog qhov pheej yig thiab zoo statin kawg tiam raws li ib tug hloov rau "Atoris", nws yog zoo dua mus rau noj ib qho piv txwv, "Merten". Qhov no yog tsis muaj tsawg kawm "Rosuvastatin" generic nrog ib tug nqi pheej yig.
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