Noj qab haus huv, Npaj
"Valium" - yog ... hauj lwm, kev qhia ntawv, kev txiav txim counterparts
"Valium" - nws yog rau cov tshuaj? Lo lus teb rau lo lus nug no koj yuav nrhiav tau ib tug me ntsis ntxiv. Peb kuj qhia koj txog yuav ua li cas no lub cuab tam tej hauj lwm, yog dab tsi cov khoom nws yog yus li nws yuav tsum tau thiab nyob rau hauv dab tsi tsim muaj.
Daim ntawv thiab muaj pes tsawg leeg ntawm ntim
"Valium" - ib tug tshuaj uas muaj peev xwm yuav yuav nyob rau hauv daim ntawv ntawm ib tug txhaj, raws li zoo li cov ntsiav tshuaj. Uas yog ib feem ntawm cov nyiaj no?
muaj 5 mg diazepam nyob rau hauv 1 mL ntawm tov rau kev txhaj tshuaj. Xws li ib tug medicament yog marketed nyob rau hauv 50 los yog 10 tsaus iav ampoules ntawm 2 ml, muab tso rau hauv cov duab los qhia thawv.
Nrog kev xav txog cov ntsiav tshuaj, lawv tej zaum yuav muaj 10 los yog 5 mg ntawm diazepam, tab sis kuj cov nram qab no ntxiv cov khoom xyaw: pob kws starch, lactose anhydrous, calcium stearate, pregelatinized starch, dyes.
Txhais tau hais tias "Valium" nyob rau hauv cov ntsiav tshuaj daim ntawv ntim rau hauv thawv ntawv, uas muaj ib tug Valium Valium.
Pharmacology ntawm cov tshuaj
"Valium" - ib tug yeeb tshuaj uas exhibits anxiolytic, miorelaksiruyuschee, sedatives, hypnotics thiab anti-qaug dab peg zog.
Ua ntej peb yuav qhia tau rau koj txog cov mechanism ntawm qhov kev txiav txim ntawm cov nyiaj, nws yuav tsum tau to taub hais tias nws yog.
Tshuaj "Valium" muaj cov nram qab no proprietary lub npe - "Diazepam". Qhov no tshuaj belongs rau cov pab pawg neeg ntawm benzodiazepines thiab muaj tseem ceeb heev nyob rau hauv cov tshuaj.
"Valium" - ib tug tshuaj uas, vim hais tias ntawm nws cov anxiolytic kev ua si, relieves nrog kev ntxhov siab vim, kev ntshai, ntxhov siab vim thiab kev nyuaj siab. Kws txawj hais tias "Diazepam" koob tshuaj-dependent ntxim rau cov central lub paj hlwb. Nyob rau hauv lwm yam lus, nyob rau hauv me me (txog 2-15 mg ib hnub twg), cov tshuaj no ua rau stimulating nyhuv, thiab loj (ntau tshaj 15 mg ib hnub twg) - ua kom loog.
nta tshuaj
Yuav ua li cas yog zoo tshaj plaws yog cov txhais tau tias raws li "Valium"? Action (central nqaij relaxant) ntawm cov tshuaj yog txuam nrog ib tug tseg polysynaptic reflexes nyob rau hauv cov leeg nrob qaum. Tau txais kev npaj no yuav ua rau ib tug txo nyob rau hauv cov ntshav siab, expansion ntawm lub coronary hlab ntsha, raws li zoo raws li txhim kho kuj mus cerebral hypoxia thiab muaj zog mob pib.
kinetics
Lub medicament "Valium" analogs uas muaj qhia hauv qab no, yog absorbed los ntawm tus mob huam (lus). Thaum zoo li no haum tshwm sim nyob rau 75% thiab lub siab tshaj plaws concentration yog mus txog tom qab 1.5 teev.
Lub lom transformation ntawm cov tshuaj nyob rau hauv lub siab. Nyob rau hauv daim ntawv no lub active metabolite nrog ib tug ib nrab-lub neej. Nyob rau hauv appointing cov tshuaj rau cov me nyuam mos cov nyhuv yog mus txog tom qab 30 teev, thiab cov neeg laus, thiab cov laus - los ntawm 100, thiab 48 cov sij hawm, ntsig txog. Nyob rau hauv no daim duab siab pathologies ntev mus rau 4 hnub.
Saib npaj muab los ntawm tib neeg lub cev tsuas yog los ntawm ob lub raum (90%) nyob rau hauv daim ntawv ntawm cov conjugates, raws li zoo raws li unchanged (2%) thiab ua ke nrog rau cov quav (8%).
zaj lus tim khawv
Nyob rau hauv dab tsi kab mob tus neeg mob tej zaum yuav muab ib tug "Valium"? Xyuas cov tub txawg qhia hais tias qhov no tshuaj yog muaj yuav tau txais nyob rau hauv cov nram no tej yam kev mob:
- chua ntawm skeletal nqaij nyob rau hauv zos kev poob plig;
- ntxhov siab vim kev ntshawv siab;
- myositis, mob caj dab, bursitis, rheumatoid plab mog-spondylitis, mob hnyav polyarthritis;
- tetanus;
- tawg, dysphoria, pais plab rwj thiab duodenum 12 (raws li ib tug ntxiv txhais tau tias), heart attack myocardial infarction;
- insomnia;
- angina;
- spastic tej yam kev mob, nrog rau cerebral palsy, mob caj dab nrog skeletal leeg nro thiab athetosis;
- lom tshuaj;
- vertebral syndrome;
- cawv tshem syndrome nrog ces xws li kev ntxhov siab vim, nro, ntxhov siab, co;
- raws li txoj cai epilepticus, kev kho mob ntawm qaug dab peg;
- psychosomatic mob nyob rau hauv Gynecology thiab Obstetrics (eg, menopausal thiab coj khaub, gestosis, mus pab txhawb zog);
- eczema thiab lwm yam kab mob uas nrog khaus thiab txob taus;
- Meniere tus kab mob ;
- hallucinatory-paranoid xeev, lub cev muaj zog excitation ntawm txawv keeb kwm (nyob rau hauv Psychiatry thiab kev kawm txoj tib neeg lub hlwb);
- ua kom tsaug zog thiab premedication (xws li, ua ntej kev phais thiab endoscopic cov txheej txheem).
Contraindications
Thaum koj yuav tsum tsis txhob siv cov tshuaj no raws li "Valium"? Cov nyhuv ntawm cov tshuaj no tsis yog tib yam li peb xav, yog tias koj txais nws:
- nyob rau hauv npau taws me ntsis;
- coma, poob siab;
- mob cawv qaug cawv;
- mob ntaub ntawv ntawm cov kab mob ntawm lub siab;
- myasthenia Heavy kev;
- lub-kaw glaucoma;
- nyob rau hauv cov me nyuam yau tshaj 6 lub hlis;
- thaum lub sij hawm lactation, thiab nyob rau hauv thawj peb lub hlis uas cev xeeb tub.
Cov tshuaj "Valium": cov lus qhia rau kev siv
Cob xam tau tias yog ib tug txhais tau tias yuav tsum yog tsuas yog ib tug tej tus kws khomob tshwjxeeb. Rau cov neeg laus cov neeg mob ib koob tshuaj ntawm cov tshuaj tom qab qhov ncauj thawj coj yuav tsum 5-20 mg ib hnub twg. Qhov no kom muaj nuj nqis ntawm cov tshuaj yog txiav txim nyob rau hauv lub heev ntawm tus kab mob cov tsos mob, raws li tau zoo raws li tag nrho cov kev soj ntsuam daim duab.
Qhov siab tshaj plaws tau koob tshuaj kho mob yog tsis ntau tshaj 10 mg. txoj kev kho thaum kawg no txhais tau tias nyob rau hauv cov ntaub ntawv ntawm kev ntxhov siab vim kev ntshawv siab yuav tsum kav txog 6 lub lis piam. Tom qab no lub sij hawm yuav tsum xa mus rau tus mus kawm tus kws kho mob, yog li ntawd nws thiaj coj ib tug yam tsawg kawg nkaus txij nkawm ntau npaum.
Lub abolition ntawm cov tshuaj twb maj suav hais tias.
Nyob rau hauv thaum muaj xwm ceev mob, active medicament yuav tsum tau muab parenterally (intramuscularly los yog intravenously). Nyob rau hauv cov ntaub ntawv no, ib koob tshuaj 2-20 mg.
Nrog tso dej Txoj kev lis ntshav ntawm cov tshuaj yuav tsum tau muab kev maj mam, ntawm ib tus nqi tsis tshaj 0.5-1 ml ib feeb.
phiv
Raws li cov kev noj tshuaj, noj nyob rau hauv saib xyuas cov tshuaj yuav ua rau ib tug kev phiv cov tshuaj tiv thaiv. Cov no muaj xws li nram qab no:
- bradycardia los yog hypotension;
- tsis concentration thiab cov tshuaj tiv thaiv tus nqi;
- yees tshuaj;
- kiv taub hau thiab mob taub hau;
- txoj kev loj hlob ntawm paradoxical tshua ntawm kev ntxhov siab vim, insomnia, hallucinations, thiab qaug dab peg;
- nco puas (luv luv);
- sab tshua ntawm lub qhov koob;
- zog mob xws li dysarthria thiab ataxia;
- kev puas tsuaj rau lub raum thiab lub siab, plab atony, tsis libido thiab potency (long-term siv cov yeeb tshuaj);
- kev tsis haum tshuaj;
- ntsoos ntsoos syndrome;
- tsis tau zoo, thiab leeg tsis muaj zog.
Nyob rau hauv lub sij hawm ntawm cov tshuaj rau tus neeg mob nws tseem ceeb heev los qhia rau nws tias qhov no yog ib tug yeeb tshuaj. Tom qab xam tau tias yog ib tug paub psychotropic neeg sawv cev tranquilizer, uas muaj ib tug xov tooj ntawm cov nyom los, cov uas tshwj xeeb tshaj yog zoo tu qab tso hom thiab ntsoos ntsoos.
Dr. designating tshuaj no yog yuam ua hauj lwm mus qhia rau tus neeg mob txog tau phiv los ntawm cov tshuaj nyob rau hauv nws lub cev, raws li zoo raws li kev lwm yam kev kho kev xaiv.
overdose ntawm cov tshuaj
Overdosing xam tau tias yog tsis kaj siab txhais tau tias nrog los ntawm xws li cov tsos mob li Cns kev nyuaj siab. Ib tug zoo xws li cov phenomenon tej zaum yuav ua heev, xws li los ntawm koj nkees nkees thiab xaus coma. Tsis tas li ntawd, thaum peb noj siab koob tshuaj ntawm cov tshuaj nyob rau hauv tus neeg mob lub tau hypotension, tsis meej pem thiab ua pa nyuaj siab.
Cov kev kho mob ntawm xws tej yam kev mob nrog rau cov proviso, yog hais tias tus neeg mob yog meej pem, yuav lub induction ntawm emesis thiab kev siv cov tshuab txais carbon. Nyob rau hauv cov ntaub ntawv uas, yog hais tias tus neeg mob tsis nco qab lawm, nws tau ntxuav los ntawm txoj kev ib plab sojntsuam, raws li zoo raws li symptomatic txoj kev kho, soj ntsuam kuaj tseem ceeb heev functions thiab cov kev taw qhia ntawm cov kua lug txhim khu diuresis.
Yuav kom ntes tus ntev ntxhov siab ntawm tus neeg mob, koj muaj peev xwm muab nws barbiturates.
Sis nrog rau lwm cov kev kho mob txhais tau hais tias
Lub medicament "Valium" ua potentiation cawv los, hypnotics, anticonvulsants, hypotensive neeg thiab antihistamines, thiab antipsychotics, general anesthetics, tricyclic antidepressants, nqaij hnaiv thiab analgesics.
Analeptic stimulants thiab yuav ho txo cov kev ua ntawm "Diazepam" tshuaj.
Antacids txo tus nqi, tiam sis tsis rau theem ntawm kev haum ntawm cov tshuaj.
Tej inhibitors ntawm microsomal oxidation li "Cimetidine", "Omeprazole" "ketoconazole" "fluoxetine" thiab "Fluvoxamine" hloov qhov tshuaj ntawm cov tshuaj nyob rau hauv kev saib xyuas, thiab kuj ua rau kom lub caij ntawm nws cov kev soj ntsuam los.
"Rifampicin" thiaj li muaj cov concentration ntawm "Diazepam" nyob rau hauv cov ntshav, thiab "Erythromycin" slows cia nws metabolism hauv lub siab.
zoo xws li cov tshuaj
Yuav ua li cas yuav hloov tau cov tshuaj no raws li "Valium"? Analogues nyob rau hauv Russia yog tsis muag nyob rau hauv pharmacies. Ntxiv mus, cov tshuaj yog tso tawm tsuas yog tom qab kev nthuav qhia ntawm kev kho mob tshuaj.
Hloov cov tshuaj tau "sibazon", "diazepam" los yog "Diapamom". Txawm li cas los, qhov no yuav tsum tau ua tsuas yog tom qab kev sib tham nrog tus kws kho mob.
Tus nqi ntawm cov tshuaj
Raws li kuv hais saum toj no, los yuav tshuaj "Valium Roche" nyob rau hauv Russia tsis tau nyob rau hauv txhua txhua lub khw muag tshuaj. Tus nqi ntawm cov tshuaj - txog ib txhiab rubles (ib pob).
Tus nqi ntawm cov nyiaj nyob rau hauv lub UK thiab lwm yam European lub teb chaws, feem ntau yog hais txog ob puas thiab tsib caug phaus ib txhiab ntsiav tshuaj (10 mg).
Yuav kom yuav nyob rau hauv lub nroog yog xws li ib tug yeeb tshuaj uas yuav ua tau raws li tag nrho cov uas yuav tsum tau muaj kev ruaj ntseg thiab zoo, kws txawj pom zoo kom siv tau rau cov tom qab, qhov twg koj yuav tau muab tas nrho cov ntaub ntawv hais txog nws txaus nyob rau hauv pharmacies thiab feem ntau ib qho kev zoo hnav.
Consumer xyuas txog cov tshuaj
"Valium" - nws yog heev nrov nrog cov neeg mob ib tug yeeb tshuaj uas yog siv raws li ib tug anxiolytic, miorelaksiruyuschego, sedatives, hypnotics, thiab anticonvulsants. Raws li cov tswv yim feem ntau ntawm cov tau txais kev pab, yog suav tias yog zoo heev tshuaj rau ntau yam kab mob, xws li, qaug dabpeg, pw tsis taus, kev ntxhov siab vim thiab thiaj li nyob. Tsis tas li ntawd noj nws yuav pab los tejzaum cov tsos mob li ntxhov siab, co thiab tshem tawm hallucinations.
Txawm li cas los, yog tsis muaj tej lub cuab tam uas yuav nplua txhua leej txhua tus. Ib txhia neeg uas siv cov tshuaj no yog tsis zoo siab. Lawv nco ntsoov tias cov tshuaj pib ua tsuas yog tom qab ib lub lim tiam. Nyob rau hauv tas li ntawd, nrog txuas ntxiv siv cov medicament ua rau ib tug loj tus naj npawb ntawm sab tshua thiab ua rau yus muaj yees ua.
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