Noj qab haus huv, Npaj
"Roxer": analogues ntawm cov tshuaj
Tshuaj "Roxer" analogs, thiab cov lus qhia rau kev siv uas peb yuav saib tom qab nyob rau hauv no tsab xov xwm, hais txog cov lipid tej tshuaj. Lawv tsa nyob rau hauv yuam cai ntawm lipid metabolism txuam nrog nce cov nqi ntawm cov lipids los yog lipoproteins nyob rau hauv cov ntshav ntshav. Qhov no mob yuav tshwm sim los ntawm ob qho tib si genetic los yog yuav kis tau, thiab nyob rau hauv kev twb kev txuas nrog asymptomatic kuaj nws yog feem ntau ntawd thaum lub sij hawm soj ntsuam kuaj cov kev tshawb cov lipid zoo.
Txais ntawm cov tshuaj yuav pab tus neeg mob kom tsis txhob muaj ib tug loj tus naj npawb ntawm loj cov kab mob thiab muaj kev noj qab nyob zoo.
Ib txhia ntawm cov tshuaj, analogs zoo
Nyob rau hauv cov tshuaj, "Roxer" cov tshuaj yog pom tias yuav ua tau heev zoo thiab ruaj ntseg. Yog li ntawd, nws yuav tsum tau muab sau tseg tias thawj zoo hloov nyob rau hauv nws daim ntawv thov yuav pom nyob rau hauv ib ob peb hnub tom qab pib ntawm kev kho mob (ntawm lub siab tshaj plaws kho nyhuv tshwm sim nyob rau hauv hais txog ib lub hlis).
Tab sis, raws li nyuab siab los ntawm cov tshuaj muaj rau "Roxer" kev qhia ntawv, tswv yim (txawm heev zoo) tsis daws tau txhua yam. Tseeb, ib co neeg mob qhov cuab tam yog tsis haum rau tej vim li cas, thiab lawv yuav tsum tig mus rau cov phooj ywg.
Nyob rau hauv xws li mob, xaiv rau tus neeg hloov tshuaj los ntawm ib tug loj daim ntawv teev cov tshuaj nrog ib tug zoo xws li cov txiav txim yuav muaj ib tug kws kho mob, thaum tej zaum los ntawm mus sib hais thiab yuam kev. Tom qab tag nrho, tej yam uas cov tshuaj thiab ntau npaum yog heev neeg.
Cov tshuaj "Roxer" chaw tsim tshuaj paus thiab analogues
Lub ntsiab active neeg sawv cev, ib feem ntawm lub "Roxer" ntsiav tshuaj - rozuvastin nws yog ib tug inhibitor (ie suppressing neeg sawv cev rau physico-tshuaj dab ..) Ntawm ib tug tshwj xeeb enzyme muab kev koom tes nyob rau hauv cov roj uas txhaws kev kawm ntawv.
Tshwj nws, ib feem ntawm cov tau piav medicament comprises:
- crospovidone, magnesium stearate,
- anhydrous lactose
- microcrystalline cellulose,
- anhydrous colloidal silica.
Tsis muaj tsawg zoo thiab muaj rau "Roxer" tshuaj analogues - tshuaj "Crestor" thiab "Atoris". Lawv muaj ib tug zoo xws li cov ntsiab cai ntawm kev txiav txim, tab sis nyob rau hauv lub xov xwm "Roxer" thiab "Crestor" ib tug thiab tib lub ntsiab active khoom sib ua zaub mov, thiab muaj cov tshuaj "Atoris" yog li ntawd yog atorvastatin.
Daim ntawv teev cov generic tshuaj "Roxer"
Nyob rau hauv tas li ntawd mus rau saum toj, cov piav statin muaj ib tug es loj daim ntawv teev cov Generics. Peb yuav sau tsuas yog cov hais tias, raws li kws txawj, yog bioequivalent, piv txwv li lawv muaj feem rau tus neeg mob lub cev yog feem ntau zoo sib xws. Yog li, feem ntau nrov tshuaj rau "Roxer" analogues nyob rau hauv Ukraine, Belarus thiab Russia - yog:
- "AKORT"
- "Klivas"
- "Roviks"
- "Rozvator"
- "Rozulip"
- "Rozart"
- "Merten"
- "Sandoz Rosuvastatin"
- "Fastrong" thiab al.
Lawv yog cov sib txawv dog dig nyob rau hauv cov nyhuv ntawm ceev: lub qeeb nyob rau hauv no hwm yog suav hais tias "Atoris", uas yog feem ntau cov tshuaj raws li ib tug tiv thaiv kev ntsuas. Tab sis rau tag nrho cov analog ntau nws yog hais tias zoo hloov yog twb pom nyob rau hauv thawj ob peb lub lim piam ntawm kev kho mob.
Nyob rau hauv ib co piv txwv, cov tshuaj "Roxer" thiab nws cov analogues
Ib yam li ntawd ntawm counterparts, thiab nyob rau feem ntau ntawm cov tshuaj "Roxer" indications rau kev siv tib yam - yog muaj cov atherosclerosis nyob rau hauv ib tug neeg mob, tus thawj, mixed los yog homozygous hypercholesterolemia, coronary mob plawv, kub siab, thiab lwm yam mob los ntawm leeg tshav kab mob.
Kws txawj ntseeg tau kom koj noj statins nyob rau hauv cov neeg mob uas muaj ib tug kev tshuaj ntsuam genetic predisposition mus cov kab mob plawv thiab hypercholesterolemia. Kom koj lub cev lipid tej tshuaj, thiab cov kws kho mob pom zoo kom cov neeg uas tsim txom lawv haus dej haus cawv thiab haus luam yeeb.
Txhua tus neeg mob koob tshuaj thiab ntev ntawm lub tshuaj kawg tus kws kho mob txiav txim ib lub zuj zus. Yog li ntawd, ib co ntawm cov neeg mob, muaj tiav zoo tau, tsis txhob noj cov tshuaj, thaum lwm tus neeg tuaj raws li ib tug tiv thaiv kev ntsuas yuav coj nws lub neej.
Yuav ua li cas yog cov kev kho mob ntawm "Roxer" npaj: cov lus qhia rau kev siv
Analogs ntawm cov tshuaj thiab cov tshuaj nws tus kheej "Roxer" ua nyob rau hauv daim ntawv ntawm cov ntsiav tshuaj uas, los ntawm txoj kev, yuav tsis faib, zom los yog zom ua ntej yuav siv. Coj lawv tsis xav txog noj mov, nqos tag nrho cov tshuaj txhaj koob tshuaj ntawm cov tshuaj nkaus thiab haus dej.
Kev kho mob txhais tau hais tias cov ntaub ntawv yeej ib txwm pib nrog ib tug tsawg koob tshuaj (10 mg ib hnub ib zaug). Nyob rau hauv cov ntaub ntawv no, nws yog kom coj mus rau hauv tus account ntau yam, xws li qhov tseeb, yog dab tsi tshuaj tus neeg mob tau txais nyob rau hauv thaum uas tig mus, raws li zoo raws li lub xeev ntawm nws lub siab thiab ob lub raum. Tom qab tswj ntawm laboratory kev ntsuam xyuas, uas yog nqa tawm txog ib lub hlis tom qab pib ntawm txoj kev kho, pib koob tshuaj yuav tau nce mus rau 20 mg. Nyob rau hauv tej rooj plaub, cov neeg mob muaj homozygous familial hypercholesterolemia, thiab koob tshuaj ntau zog rau 40 mg. Incidentally, qhov kev siv ntawm high-koob tshuaj "Roxer" tshuaj yuav tsum tau tas li xyuas ntawm tus neeg mob tus mob.
Raws li taw tes qhia tawm los ntawm cov kev qhia ntawv mus rau yeeb tshuaj, rau nws cov ntau dua efficiency yog tsim nyog them sai sai tsis tsuas mus rau lub concentration ntawm triglycerides thiab roj uas txhaws taus tus neeg mob, tab sis kuj nyob rau hauv nws muaj hnub nyoog, poj niam txiv thiab haiv neeg. Qhov no yog vim lub fact tias lub concentration ntawm cov tshuaj, nyob ntawm seb lub saum toj no tsis tej zaum yuav txawv - piv txwv li, Isdias Asmesliskas thiab Mongoloid saum toj no nws, thiab chaw pib lub noj tshuaj npaum cas yuav tsum tau rau nws rov qab, yuav tsum tau ntau tshaj li nyob rau hauv Caucasians.
Contraindications rau kev siv ntawm "Roxer" npaj
Raws li hais saum toj no, cov tshuaj yuav tsum tau muab los ntawm koj tus kws kho mob. Qhov tshwj xeeb siv sij hawm mus rau hauv tus account lub fact tias thaum lub sij hawm exacerbations ntawm daim siab tus kab mob thaum lub sij hawm cev xeeb tub thiab lactation, thiab nyob rau hauv mob loj heev raum insufficiency tshuaj "Roxer" los yog nws analogues yog tsis muab.
Txhob lawv thiab cov neeg mob neuromuscular cov kab mob (nyob rau hauv particular, nrog myopathy), cov neeg mob ib txhij tau txais raws li ib tug antidepressant "Tacrolimus", cov poj niam uas deev muaj hnub nyoog uas tsis siv contraceptives, raws li zoo li cov me nyuam nyob rau hauv kaum yim xyoo ntawm lub hnub nyoog, thiab cov neeg laus tom qab 70 xyoo.
Npe txaus ntshai npau taws me ntsis neeg sawv cev nyob rau hauv ib ntsiav tshuaj Cheebtsam.
phiv
Tshuaj "Roxer" analogues ntawm no txhais tau tias - lawv ua tau tag nrho cov ua raws li ib tug tshwm sim ntawm cov kev phiv. Lawv yuav tsum tau ntaus nqi feem ntau ib tug tsis haum cov tshuaj tiv thaiv mus rau yeeb tshuaj, uas yog manifested nyob rau hauv daim ntawv ntawm cov khaus, daim tawv nqaij ua pob liab vog, thiab urticaria, kom txog rau thaum txoj kev loj hlob ntawm angioedema.
Tshwm sim nyob rau hauv cov neeg mob uas gastrointestinal mob thiab kev khiav dej num, uas yog qhia los ntawm mob plab, xeev siab thiab, nyob rau hauv uas tsis tshua muaj mob, ntuav. Kaw thiab tus neeg mob ntawm pancreatitis, mob ntawm hauj lwm ntawm skeletal leeg, feem ntau tshwm sim li myalgia (mob leeg) los yog tsawg dua - myopathy thiab qaug zog phenomena.
Muaj mob ntawm ob lub raum thiab lub mob txeeb zig, nrog los ntawm ib tug nce nyob rau hauv tus nqi ntawm cov protein nyob rau hauv cov zis.
Thaum muab "Roxer" cov tshuaj yuav tsum tau coj mus rau hauv tus account thiab tseem los ntawm cov kuaj tsis. Yuav ua rau kom cov kev ua ntawm creatine kinase, hloov lub concentration ntawm qab zib los yog bilirubin, thiab cov thyroid hormones.
tau overdose
Yog hais tias koj ntau tshaj qhov kws koob ntawm cov tshuaj yog ua tau rau overdose "Roxer". Cov chaw tsim tshuaj paus ntawm cov tshuaj no nyob rau ntawm no qhia ntau txog kev uas nyob rau hauv ib txais tsa koob tshuaj clinically yam ces overdose yog tsis cai.
Nyob rau hauv cov ntaub ntawv ntawm tej yam tshwm sim ntawm toxicity rau tus neeg mob yog muaj symptomatic kev kho mob thiab txhawb nqa txoj kev kho. Pom zoo thiab ntxiv xyuas ntawm daim siab kev ua, raws li tau zoo raws li creatine kinase kev ua si.
Los ntawm tau txais lipid tej tshuaj yuav tsum tau npaum li cas tiag!
Kev npaj "Roxer" (xws li analogs) tsis muaj feem xyuam rau lam cov khoom npaj rau nws tus kheej-thawj coj. Lawv yuav tsis Iwj, nyob rau hauv ib tug maj "coj lub cholesterol," raws li nws nkawd frivolous rau ib co neeg mob. Yog li ntawd, lipid tej tshuaj muaj tsuas los ntawm cov tshuaj, thiab kev kho mob yog nqa tawm los ntawm lawv nyob rau hauv ib tug neeg txhaj koob tshuaj thiab qhov kuaj tswj tau.
Yog hais tias tus neeg mob tau muab cov ntsiav tshuaj "Roxer" los yog lawv sib npaug, nws yuav tsum xyuas nrog koj tus kws kho mob, tej kev phiv los yuav tsum ceev faj ntawm yuav ua li cas coj thaum lawv tshwm sim, qhia kom meej lub sij hawm uas tus me nyuam ntawm cov ntshav mus rau lub tswj thiab thiaj li nyob. N.
Tsuas yog thaum cov tej yam kev mob yog statins tej zaum yuav txhais tau tias ho sim haum tus neeg mob lub neej thiab tau txhawb nws cov kev kho mob.
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