Noj qab haus huv, Npaj
Antidepressant "Velaksin": tus neeg mob testimonials, cov lus qhia rau kev siv, analogs
Kuv yuav antidepressants tsis muaj ib tug tshuaj? Ib daim ntawv teev tej khoom yog tsis loj. Qhov no yog vim lub fact tias lawv muaj peev xwm yuav hom, thiab ib tug tswv tsev ntawm sab los. Yog li ntawd, ua ntej noj xws txhais tau tias, yuav tsum mus ntsib ib tug tshwj xeeb.
lus qhia dav dav
Kev nyuaj siab yog tsis kho los ntawm cov tshuaj. Tab sis los txhim kho lub hauj lwm ntawm lub paj hlwb, cov kws kho mob ntau tseem muab rau lawv cov neeg mob ntau yam antidepressants. Ib tug ntawm lawv yog cov tshuaj "Velaksin". Testimonials txog qhov cuab tam thiab nws cov nta thiab cov lus qhia rau kev siv yuav tsum hais hauv qab no.
Muaj pes tsawg leeg ntawm yeeb tshuaj, nws daim ntawv ntawm ntau lawm
Nyob rau hauv dab tsi daim ntawv nws ua ib antidepressant li "Velaksin"? Ntsiav tshuaj thiab tsiav tshuaj - yog tib cov neeg ntaub ntawv ntawm qhov kev siv yeeb tshuaj.
Ntsiav tshuaj "Velaksin" yog dawb, engraved rau ntawm ib sab "E741", thiab ib tug yeej tiaj tus zoo thiab chamfer. Lawv active ingredient yog venlafaxine, uas yog sawv cev nyob rau hauv daim ntawv ntawm ib tug hydrochloride. Tsis tas li ntawd muaj nyob rau hauv cov tshuaj no muaj xws li koom haum pab Cheebtsam xws li colloidal silica anhydrous, lactose monohydrate, sodium cov hmoov txhuv nplej glycolate, magnesium stearate thiab MCC.
Uas ntsiav tshuaj nyob rau hauv sawv hlwv packs thiab cartons feem.
Tshuaj "Velaksin" - tsiav tshuaj, cov lus qhia rau kev siv uas yog nrog rau hauv lub ntim, daim ntawv, gelatin thiab khoom. Lawv muaj txiv kab ntxwv-daj hau thiab ib tug tsis muaj kob substrate. Lub active tivthaiv ntawm daim ntawv no tseem yog ib tug compound venlafaxine. Nyob rau hauv tas li ntawd mus rau nws lub muaj pes tsawg leeg ntawm cov tshuaj no muaj xws li ntxiv cov khoom xyaw.
Raws li cov tshuaj ua hauj lwm zoo?
"Velaksin" - ib tug tshiab tiam ntawm anti-depressant. Raws li cov tshuaj qauv ntawm nws cov active tshuaj tsis yog rau tej lub npe hu chav kawm ntawv ntawm antidepressants (e.g., tricyclic, tetracyclic, los yog lwm yam). Kws txawj hais tias cov tshuaj yog active enantiomer 2 racemate.
Lub hauv paus ntsiab lus ntawm kev txiav txim ntawm cov tshuaj no yog hais txog nws lub peev xwm rau potentiate lub Cns paj impulse kis tau tus mob.
Raws li cov lus qhia, venlafaxine thiab nws loj metabolite (EFA los yog O-desmetilvenlafaksin) sawv cev hwj chim inhibitors ntawm lub reuptake ntawm norepinephrine thiab serotonin thiab tsis muaj zog inhibitors ntawm dopamine reuptake. Peb tsis tau hais tias cov tshuaj yog tau txo tus beta-adrenergic ua si tom qab ib tug hluas thiab qhov tshuaj. EFA thiab venlafaxine yog Attendance zoo tiv thaiv reuptake ntawm neurotransmitters.
Yuav ua li cas lwm tus neeg yog zoo kawg li tshuaj "Velaksin"? Phau Ntawv Qhia hais tias lub active ingredient ntawm cov tshuaj muaj ib qho kev sib ze nrog rau cov n- thiab m-cholinergic receptors, lub hlwb α1-adrenoceptors thiab histamine H1-receptors. Tsis tas li ntawd, nws cheeb qhov uas cov kev txiav txim ntawm Mao thiab twb tsis muaj kev zoo sib thooj nrog fentsiklidinovymi, opioid, benzodiazepine thiab NMDA-receptors.
Lub kinetics ntawm cov tshuaj
seb cov tshuaj yog absorbed, "Velaksin" (ntsiav tshuaj)? Cov lus qhia rau Siv hais tias lub active tivthaiv ntawm cov tshuaj no yog zoo heev absorbed los ntawm lub plab. Tom qab ib tug tib koob tshuaj medicament nyob rau hauv ib tug ntau npaum ntawm 25-150 mg ntawm nws siab tshaj plaws nyob rau hauv concentration cov ntshav yog mus txog tom qab 2.4 teev. Yog li venlafaxine yog feem metabolized thaum lub sij hawm thawj pass los ntawm lub siab. Yog hais tias cov tshuaj yog noj nrog zaub mov, thaum nws ncov concentration nce los ntawm 27-30 feeb nyob rau hauv ntshav.
Lub ntsiab metabolite yog suav tias yog ib tug txhais tau tias ntawm O-desmetilvenlafaksin. Nws ib nrab-lub neej thiab tshem tawm ib nrab-lub neej ntawm venlafaxine yog 11 thiab 5 teev, feem (tso zis nyob rau hauv unchanged daim ntawv los ntawm lub ob lub raum).
Lub kinetics ntawm cov tshuaj nyob rau hauv tshwj xeeb soj ntsuam lub sijhawm
Tshuaj "Velaksin" qhia no yuav tsum tau nyeem nyob rau hauv cov neeg uas muaj mob npuas paug ntawm lub siab muaj lwm yam kev tig tau nta. ntshav concentration ntawm cov tshuaj muaj zog nyob rau hauv cov neeg mob, thiab nws tus nqi ntawm feem, on qhov tsis tooj, txo.
Rau hauv loj heev raum insufficiency, raum tsis ua hauj lwm thiab hauj sim tag nrho clearance EFA thiab venlafaxine yog txo kom tsawg thiab cov tshem tawm ib nrab-lub neej lub sij hawm yog lengthened.
Nws yuav tsum tau muab sau tseg tias tus tub los ntxhais thiab muaj hnub nyoog ntawm tus neeg mob tsis cuam tshuam rau tshuaj ntawm cov tshuaj nyob rau hauv kev saib xyuas.
indications rau
Vim li cas peb yuav tsum tau ib lub cuab tam xws li "Velaksin"? Kev siv cov tshuaj no muaj nyob rau hauv lub kev nyuaj siab ntawm ntau yam keeb kwm (rau cov kev kho mob thiab prophylaxis).
Bans lub sij hawm
Nyob rau hauv dab tsi tej yam kev mob yuav tsis siv cov tshuaj "Velaksin"? Xyuas ntawm cov neeg mob thiab cov kws kho mob hais tias cov tshuaj no yog txhob tau txais:
- thaum uas tau txais Mao inhibitors ;
- nyob rau hauv kev mob loj raum mob;
- thaum lub sij hawm ib tug txhawj los yog tsim cev xeeb tub;
- nyob rau hauv kev mob loj mob ntawm lub siab;
- thaum lub sij hawm pub niam mis;
- nyob rau hauv kev ua hluas thiab thaum yau, uas yog, kom txog thaum lub hnub nyoog ntawm feem ntau;
- nrog siab rhiab heev mus rau yeeb tshuaj.
Tsis tas li ntawd, qhov no tshuaj yuav tsum tau ua tib zoo coj nyob rau hauv tsis ruaj tsis khov angina, heart attack myocardial infarction (nrog rau cov tshiab khiv migrated), kub siab, convulsions keeb kwm, tachycardia, poob phaus, nce intraocular siab, lub kaum ntse ntse-kaw glaucoma, predisposition mus los ntshav los ntawm txheej thiab daim tawv nqaij, manic lub xeev.
Tshuaj "Velaksin" (ntsiav tshuaj): cov lus qhia rau kev siv
Antidepressant "Velaksin" yuav tsum tsuas yog noj thaum lub sij hawm ib tug noj mov. Cov pom zoo starting koob tshuaj ntawm cov tshuaj yog 75 mg, muab faib nyob rau hauv 2 faib koob tshuaj (i.e., 37.5 mg ib hnub ob zaug), txhua txhua hnub.
Yog hais tias tom qab ob peb lub lim piam ntawm txoj kev kho, tus neeg mob tus mob tsis tau zoo tuaj, txhua hnub koob tshuaj yog nce rau 150 mg ib hnub twg, nyob rau hauv ob faib koob tshuaj (i.e., 75 mg ib hnub ob zaug).
Yog hais tias tus neeg mob yuav tsum tau ib tug ntau dua koob ntawm ib tug antidepressant (e.g., loj depressive teeb meem, los yog lwm yam tej yam kev mob uas yuav tsum tau txoj kev kho ruaj ruaj), ces tus ti teg taw yuav xaiv 150 mg ntawm yeeb tshuaj nyob rau hauv 2 teev, thiab ces maj mam nce lub koob tshuaj los ntawm 75 mg (2-3 hnub tom qab ntawd) mus cuag tej yam tshwm sim.
Raws li cov lus qhia, lub siab tshaj plaws ntau npaum "Velaksina" yog 375 mg ib hnub twg. Tom qab tau zoo lub Desired nyhuv, nws muaj peev xwm yuav maj mam txo qis rau qhov tsawg kawg nkaus theem.
Relapse kev tiv thaiv thiab txij nkawm txoj kev kho
Kev tu ntawm cov nyiaj yuav muab tau rau lub hlis. Nyob rau hauv cov ntaub ntawv no, cov tshuaj noj nyob rau hauv tsawg heev koob tshuaj.
Nyob rau hauv me me raum insufficiency kho dosing regimen yog yuav tsum tau. Nyob rau hauv ib tug zoo li tus kab mob loj tsawv koob tshuaj pom zoo sab by 25-50%. Nws yuav tsum tau muab sau tseg tias venlafaxine yuav tsum tsis txhob yuav siv nyob rau hauv mob loj heev raum insufficiency, vim tsis muaj ntaub ntawv nyob rau hauv kev ruaj ntseg ntawm xws txoj kev kho rau hnub tim, tsis muaj.
Cov neeg uas yog nyob rau hauv hemodialysis, yuav tsum tau txais 50% ntawm lub niaj zaus txhua txhua hnub ntau npaum ntawm cov tshuaj tom qab qhov kev sib kho xaus.
Rau me ntsis hepatic insufficiency kho dosing regimen kuj tsis yuav tsum tau. Thaum tus kab mob no yog ib sim koob tshuaj yuav tsum raug txo los ntawm 50%. Nrog hais txog mus rau mob hnyav hepatic tsis ua hauj lwm, nyob rau hauv rooj plaub no tus siv venlafaxine yog txwv tsis pub.
Nyob rau hauv cov neeg laus, cov tshuaj "Velaksin" yuav tsum tau siv nrog huab ceev faj. Qhov no yog vim cov tau ua txhaum ntawm lub ob lub raum. Cov neeg mob yuav tsum muab tus nqi qis tshaj zoo koob. Nyob rau hauv cov ntaub ntawv no, tus neeg mob yuav tsum tau nyob rau hauv qhov kev kho mob saib xyuas.
Ncua tseg antidepressant
Thaum kawm tiav ntawm tau txais cov tshuaj yuav tsum tau suav hais tias yuav tau cov tshuaj maj (nyob rau hauv ib lub lim tiam). Nws yuav tsum tau mus soj ntsuam cov mob ntawm tus neeg mob, nyob rau hauv thiaj li yuav txo tau txoj kev pheej hmoo ntawm kev phiv tshuaj txuam nrog rau abolition ntawm cov tshuaj.
Lub sij hawm yuav tsum tau rau lub teb cessation ntawm cov tshuaj, nyob rau hauv lub tshuaj, ntev ntawm txoj kev kho thiab ib tug neeg rau ib tug neeg.
phiv
Yuav ua li cas yog cov pliaj los ntawm cov tshuaj yuav ua rau "Velaksin"? Testimonials hais tias txoj kev loj hlob ntawm cov neeg los yog lwm yam kev phiv cov txheej xwm nram qab no siv ntawm no lub cuab tam nyob rau hauv lub koob tau txais.
Qhov feem ntau heev tshua manifested tsis zoo xwm muaj xws li cov nram qab no:
- tawg, tsis qab los noj mov, txawv txav kev npau suav, cem quav, insomnia, xeev siab, kais ntawm daim tawv nqaij, tshee, ntuav, mob tu-sauv, qhov ncauj qhuav;
- hallucinations, kab mob siab, poob phaus, tachycardia, hyponatremia, apathy, postural hypotension, kiv taub hau, manic cov tshuaj tiv thaiv, lub paj hlwb excitability, yawning, paresthesia, neuroleptic syndrome, stupor, serotonergic syndrome;
- nce nqaij laus, qaug dab peg, dysuria, photosensitivity, urinary tuav, anorgasmia;
- los ntshav nyob rau hauv daim tawv nqaij, txawv txav ejaculation, menorrhagia, tsis libido, tawm hws;
- thrombocytopenia, kev pab cuam tshuam, kev erythema multiforme, mydriasis, Stevens - Johnson, pom tau qhov sib cuam tshuam, impaired saj, prolongation ntawm los ntshav lub sij hawm, tsis muaj zog, daim tawv nqaij ua pob liab vog, nkees, anaphylactic tshua.
tswv yim pom zoo
Muag seb antidepressants tsis muaj ib tug tshuaj? Ib daim ntawv teev cov tshuaj no yog tsis heev loj ( "Prozac", "Paxil", "Despres", "Azafen", "Persian", "amitriptyline"), thiab cov tshuaj "Velaksin" yog tsis muaj nyob rau hauv nws. Yuav nyob rau hauv pharmacies, koj ua tau tsuas yog los ntawm tus kws kho mob tshuaj.
Ua ntej yuav noj cov tshuaj no nyob rau hauv kev ntsuam xyuas, tshwj xeeb tshaj yog cov neeg mob uas depressive ntshawv siab, yuav tsum tau suav hais tias ib siab yuav qhov muaj tseeb ntawm suicidal npaj siab. Nyob rau hauv no hais txog, thaum pib ntawm yeeb tshuaj kho pom zoo rau siv nyob rau hauv qhov tsawg kawg nkaus koob thiab nyob rau hauv ze kho mob saib xyuas.
Cov neeg uas muaj ob peb vas ntshawv siab thaum lub sij hawm kev kho mob nrog antidepressants tej zaum yuav tsim manic los yog hypomanic lub xeev.
Cov neeg mob yuav tsum tau mus ceeb toom rau ntawm qhov yuav tsum tau kom sai li sai pom ib tug kws kho mob nyob rau hauv cov ntaub ntawv ntawm urticaria hais, ua pob ua xyua los yog tsis haum.
Ib txhia neeg nyob rau hauv tus txheej txheem ntawm tau txais venlafaxine cai ib koob tshuaj-dependent nce nyob rau hauv cov ntshav siab.
Cov laus cov neeg mob yuav tsum tau ceeb toom ntawm ib tug ua tau ua txhaum ntawm lub siab uas tshuav nyiaj li thiab kiv taub hau kev loj hlob.
Thaum lub sij hawm kev kho mob ntawm cov nyiaj yuav tsum tsis txhob noj haus.
Antidepressant "Velaksin": tus neeg mob testimonials, khoom analogues
Yuav ua li cas cov neeg no hais txog cov tshuaj no rau ib tug neeg mob? Muaj ntau cov kev pab muaj qhia txog ib tug loj tus naj npawb ntawm cov kev phiv uas tshwm sim thaum noj tshuaj no. Heev feem ntau cov tshuaj no ua rau kev phiv tshuaj xws li nkees nkees, tsis muaj zog, insomnia, mob chua leeg, txawv txav xav, kev nyuaj siab thiab tsis meej pem. Nyob rau hauv tas li ntawd, ib co neeg mob hais tias cov no los nyob twj ywm tom qab kawm tiav ntawm kev kho mob. Tsis tas li ntawd, ntau cov neeg siv tsis txaus siab txog cov tsos ntawm ntsoos ntsoos cov tsos mob thiab dependence.
Yuav ua li cas yuav hloov tau antidepressant xws li "Velaksin"? Analogs ntawm cov tshuaj no yog tsis muaj nyob rau hauv tag nrho cov drugstores. Raws li txoj cai, kws txawj Cov no muaj xws li nram qab no: "Venlafaxine Sandoz", "Efevelon", "Alvent", "Nyuvelong", "Velafaks", "Dapfiks", "Voksemel", "Venlaksor", "Vensuert", "venlafaxine".
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