Noj qab haus huvNpaj

"Metadoksil": xyuas quav dej quav cawv, cov lus qhia rau kev siv, muaj pes tsawg leeg thiab cov hauj lwm

Yuav ua li cas zoo behaves tshuaj "Metadoksil"? Xyuas ntawm quav dej quav cawv, tus nqi ntawm cov khoom no thiab nws cov indications yuav sib tham txog hauv qab no. Tsis tas li ntawd nyob rau hauv no tsab xov xwm, koj yuav kawm tau txog txoj kev ntawm daim ntawv thov ntawm cov tshuaj, nws tshwm sim thiab contraindications.

Hauj lwm, daim ntawv, muaj pes tsawg leeg

Tshuaj "Metadoksil" (quav dej quav cawv kev xyuas txog nws yuav tsum tau qhia rau hauv qab no) yog muaj rau cov muag khoom nyob rau hauv cov nram no cov ntaub ntawv:

  • Biconvex, puag ncig dawb ntsiav tshuaj nrog Valium rau ntawm ib sab thiab engraved nrog lub npe ntawm cov khoom - nyob rau lwm yam. Nws active ingredient yog L-ob pyridoxine pyrrolidone carboxylate-tsib los yog hu li ntawd metadoksin. Tsis tas li ntawd nyob rau hauv qhov cuab tam yog lub MCC thiab magnesium stearate.
  • Lub ntshiab tov cov kev txhaj tshuaj yog tsis muaj kob los yog yellowish tint. Nws lub ntsiab tivthaiv no kuj metadoksin. Sib nrug los ntawm nws, nyob rau hauv cov tshuaj muaj pes tsawg leeg muaj xws li sodium edetate, dej d / thiab sodium metabisulfite thiab methyl parahydroxybenzoate.

nyhuv ntawm cov tshuaj

"Metodoksil" - ib tug kho rau alcoholism. Nws kuj yog ib tug txhais tau tias ntawm uas qhia detoxification thiab hepatoprotective zog.

Hepatoprotective nyhuv ntawm cov tshuaj vim nws daim nyias nyias stabilizing nyhuv. Nyob rau hauv tas li ntawd, cov tshuaj no muaj peev xwm sawv ntawm kev txo tus piv ntawm free unsaturated thiab nyeem fatty acids. Raws li ib tug tshwm sim uas muaj zog kuj rau cov teebmeem ntawm hepatocyte peroxidation ntawm cov nqaijrog sawv nyob rau hauv tus ntawm tshuaj lom tshuaj mas siv.

Detoxification thaj chaw ntawm cov tshuaj vim qhov ua kom daim siab enzymes uas muab kev koom tes nyob rau hauv lub metabolism ntawm ethanol (nyob rau hauv particular cawv dehydrogenase thiab acetaldehyde dehydrogenase), ho accelerates tus txheej txheem ntawm nws cov tshem tawm ntawm lub cev thiab, raws li ib tug tsim nyog tau, nws thiaj li cov tshuaj lom nyhuv.

nta tshuaj

Yuav ua li cas yog zoo tshaj plaws tshuaj "Metadoksil"? Instruction kev hais tias nws active tshuaj tiv thaiv lub tsim ntawm hais xws li collagen thiab fibronectin, thiab tiv thaiv lub hnab khib triglycerides, uas ho slows txoj kev loj hlob ntawm mob npuas paug.

Nws yuav tsum tau muab sau tseg tias qhov cuab tam yog tau kom lub sij hawm ntawm nyem ntawm ntsoos ntsoos cov tsos mob, txo lub Somatic thiab puas siab puas ntsws tsos mob ntawm dej cawv tshem syndrome.

Peb tsis tau hais tias metadoksin activates GABA-ergic thiab cholinergic neurotransmitter system tsis pub lub cev muaj zog excitation, pab txoj kev luv luv nco thiab xav. Nyob rau hauv tas li ntawd, ib yam khoom uas muaj peev xwm sawv ntawm exerting ib nonspecific anxiolytic thiab antidepressant los, raws li zoo raws li tau kom tsis txhob yees rau haus dej haus cawv.

kinetics

Tom qab noj cov tshuaj hauv nws yog sai absorbed los ntawm cov hnyuv. Metadoksin muaj ib tug high bioavailability (kwv yees li 60-85%). Nws ruaj rau ntshav cov nqaijrog 50%.

Qhov no feem yog metabolized nyob rau hauv lub siab mus rau daim ntawv active derivatives - pyrrolidone carboxylate thiab pyridine.

Ib nrab-lub neej tshuaj los ntawm parenteral thawj coj los yog haus ntawm 45-57 feeb. Kwv yees li 40-50% ntawm cov tshuaj zoo nkaus li nyob rau hauv cov zis thaum lub sij hawm lub hnub thiab txog 35-50% - nyob rau hauv cov quav hauv 95 teev.

zaj lus tim khawv

Nyob rau hauv dab tsi tej yam kev mob qhov zoo tshaj tshuaj behaves "Metadoksil"? Xyuas quav dej quav cawv hais tias qhov no tshuaj yog zoo heev rau:

  • alcoholism;
  • nyob rau hauv cov kev kho mob ntawm daim siab tus kab mob, nrog rau dej etiology;
  • cawv tshem syndrome ;
  • cawv qaug cawv, xws li mob.

Contraindications

Saib cov tshuaj yog ua rau:

  • kev pub niam mis;
  • hnub;
  • siab rhiab heev rau lub ntsiab ntawm cov tshuaj.

Nrog kev saib xyuas lub tsev no yuav tsum tau siv nyob rau hauv Parkinson tus kab mob, tshwj xeeb tshaj yog yog hais tias tus neeg mob yog twb siv levodopa. Qhov no yog vim lub fact tias metadoksin tau txo cov hauj lwm zoo ntawm lub yav tas.

Tshuaj "Metadoksil": cov lus qhia rau kev siv

Xyuas qhia tias kev siv ntawm cov nyiaj yuav tsum tsuas yog tom qab kev sib tham nrog ib tug tshwj xeeb.

Thaum haus cawv qaug cawv, tshwj xeeb tshaj yog mob, active tshuaj yog muab intramuscularly nyob rau hauv ib tug ntau npaum ntawm 300-600 mg los sis intravenously - 300-900 mg.

Thaum muab intravenously, cov tshuaj txhaj koob tshuaj qhia yav tas los diluted nyob rau hauv 5% dextrose tov los nrog 500 ml ntawm sodium tshuaj dawb. Nyob rau hauv xws daim ntawv cov kev npaj yog tswvcuab dropwise, tshaj 1.4 teev.

Raws li ib feem ntawm ib tug ua ke kev kho mob ntawm daim siab kab mob, thiab mob alcoholism lub cuab tam 500 mg rau noj ib hnub ob zaug rau 25-35 feeb ua ntej noj mov. Qhov no koob tshuaj yuav tau nce mus rau 500 mg peb zaug ib hnub twg.

Hoob no ntawm txoj kev kho nrog cov tshuaj no yuav tsum kav tsawg kawg yog 90 hnub.

Thaum abstinent syndrome (dej) lub medicament yog xeem intravenously los ntawm Txoj kev lis ntshav ntawm ib koob tshuaj 900 mg ib zaug ib hnub twg rau 3-7 hnub (nyob ntawm seb tus neeg mob).

phiv

Yuav ua li cas tsis zoo kev txiav txim yog tshuaj "Metadoksil"? Xyuas ntawm quav dej quav cawv tau qhia hais tias nyob rau hauv lub ntsiab lus teb ntawm kev thov no txhais tau tias lawv feem ntau tsim kev tsis haum tshuaj loj.

Nws yuav tsum tau muab sau tseg tias cov neeg bronchospasm zaum yuav tshwm sim nrog bronchial hawb pob (ntau zaus yog tias koj siv tshuaj).

tej ntaub ntawv

Cov tshuaj rau "Metadoksil" txhaj muaj ib tug tivthaiv xws li sodium metabisulfite. Qhov no cov ntaub ntawv uas yuav ua rau muaj mob hawb pob nyob rau hauv raug neeg kev tsis haum tshuaj, raws li zoo raws li lawv amplification.

Tshuaj "Metadoksil": xyuas quav dej quav cawv

Tu siab, txheeb xyuas ntawm "Metadoksil" npaj, muaj yog tsis heev npaum li cas. Txawm li cas los, ntawm cov neeg uas tshuav cov neeg nws mus alcoholism, peb yuav xyuam xim xaus tias cov tshuaj muaj ib tug zoo zoo nyob rau hauv cov kev kho mob ntawm cov cawv dependence.

Raws li rau cov hauj lwm zoo ntawm kev kho mob ntawm ntsoos ntsoos cov tsos mob, tus neeg mob tawm tswv yim yog markedly divergent. Ib txhia sib ceg hais tias yog xws li ib tug lub xeev tshuaj pab zoo heev, thaum lwm tus neeg - tsis tau pom tej nyhuv.

Kuj nrhiav tau ib tug ntau ntawm tsis zoo txog tus nqi ntawm no lub cuab tam. Raws li ib tug txoj cai, nws yog 1250-1450 rubles.

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