Noj qab haus huv, Npaj
"Amlodipine": dab tsi pab, cov lus qhia rau kev siv, analogs, xyuas
Yuav ua li cas yog tawg? Lo lus teb rau lo lus nug no yog paub tias yuav muaj coob tus neeg, tshwj xeeb yog cov neeg laus. Raws li koj paub, qhov no yog ib tug pheej nce nyob rau hauv cov ntshav siab, nyob rau hauv uas lub cai ntsuas xws li 150/90 mmHg. Art. thiab saum toj no.
Nws yog ntseeg hais tias tawg yog feem ntau tus kab mob ntawm cov hlab plawv system. Pheej nce nyob rau hauv cov ntshav siab yog cai nyob rau hauv 25-30% ntawm cov neeg laus cov pejxeem. Los ntawm txoj kev, muaj hnub nyoog yog ib tug kab mob pom nyob rau hauv 55-65% ntawm cov neeg.
Yog vim li cas muaj yog tawg? Qhov no tshwm sim yuav tshwm sim vim muaj ntau yog vim li cas. Feem ntau cov feem ntau nyob rau hauv cov neeg laus lub siab ntawm lub nce raws li ib tug tshwm sim ntawm lub psycho-lub siab lub ntsws lim. Yog li ntawd cov neeg nws mus tawg, yuav tsum tau raws li siab tus tus.
Peb tsis tau hais tias tus kab mob no feem ntau tshwm sim vim muaj ib tug sedentary txoj kev ua neej, hnub nyoog, poj niam txiv (ntau ntau nyob rau hauv lub fairer ib nrab ntawm cov tib neeg), ntev ntsev kom tsawg, gipokaltsievoy noj cov zaub mov, dej caw, caj, rog, haus luam yeeb, mob ntshav qab zib thiab t. d.
Yog nws tsim nyog los kho tawg? Cov kws kho mob hais tias yog hais tias koj xav tias unwell, cov neeg mob yuav tsum tau noj tshuaj uas txo cov ntshav siab. Rau ib tug ntawm lawv nqa ib tug yeeb tshuaj raws li "Amlodipine". Tshwm sim los ntawm qhov cuab tam, nws cov nta, raug nqi, thiab analogs muaj li nram no.
Hauj lwm ntawm lub lam khoom, nws muaj pes tsawg leeg thiab packing
Nyob rau hauv dab tsi daim ntawv no yog manufactured tshuaj "Amlodipine", tus nqi ntawm uas yog teem tawm hauv qab no? Xam tias yog ib tug yeeb tshuaj ua nyob rau hauv daim ntawv ntawm cov dawb thiab ploskotsilindricheskoy daim ntawv ntsiav tshuaj. Nws tam sim no caij yog amlodipine.
Qhov no formulation yog muag nyob rau hauv lub cell contour (10 ntsiav tshuaj) uas yog tau ntim rau hauv cartons.
Lub mechanism ntawm qhov kev txiav txim ntawm cov tshuaj
Yuav ua li cas zoo yog "Amlodipine"? Raws li cov lus qhia, cov tshuaj exhibits ib tug qhia antihypertensive thiab antianginal zog. Tsis tas li ntawd, nws tsis muab calcium ions kom penetrate lub membrane ntawm myocardial hlwb thiab leeg tshav hlwb.
Yuav ua li cas yog cov tshuaj "Amlodipine"? Los ntawm dab tsi pab no tshuaj? Nws yog zoo thiaj li ntshav siab. Qhov no yog vim cov tshuaj muaj peev xwm los nthuav cov hlab ntsha.
Nws yuav tsum tau muab sau tseg tias pom tau hais tias cov tshuaj exhibits ib antianginal nyhuv. Qhov no cov khoom teejtug uas tshuaj no yog muab los ntawm nws tam sim no lub caij. Cov kws kho mob tau qhia hais tias amlodipine tsis tau tsuas yog nthuav cov arterioles (peripheral), tab sis kuj txo peripheral vascular kuj. Wherein hais tias muaj tsis ua tachycardia (reflex).
Yuav ua li cas yog cov kev tshwm sim ntawm kev siv cov tshuaj "Amlodipine"? Nyob rau dab tsi ua rau qhov cuab tam? Tsaug rau cov tshuaj no ib tug neeg muaj lub siab pib haus tsawg heev zog thiab ho txo myocardial oxygen thov.
Kinetics ntawm yeeb tshuaj
Tshuaj "Amlodipine" lub siab (siab) yog absorbed los ntawm cov hnyuv heev maj mam, tab sis nyob rau hauv nws txoj kev paub. Lub ncov concentration ntawm nws active muaj nyob rau hauv cov ntshav yog mus txog tom qab 8.5 teev. medicament Ntshav protein losis tswvyim dabtsi yog kwv yees li 98%.
Lub medicament "Amlodipine", uas txiav txim yog raws kev coj kom siab yuav txo tau, undergoes tsawg heev metabolism. Nyob rau hauv daim ntawv no derivatives uas muaj ib tug tsis tshua muaj pharmacological kev ua si. Metabolized tshuaj thaum dhau los ntawm lub siab.
Qhov nruab nrab ib nrab-lub neej ntawm amlodipine thiab nws cov derivatives yog 36 xuab moos. Thaum xav tsa cov ntshav siab yog ib lub sij hawm yuav muab ntau zog mus txog ob hnub, cov neeg laus - mus txog rau 66 teev, thiab daim siab tsis ua hauj lwm - mus txog rau 58 teev.
Muab tshuaj nyob rau hauv daim ntawv ntawm cov metabolites los ntawm cov hnyuv thiab ob lub raum.
Tshuaj "Amlodipine": dab tsi pab?
Nyob rau hauv tej rooj plaub, tshuaj tej zaum yuav muab suav hais tias yuav tsum tau muab rau tus neeg mob? Indications rau lub txais tos ntawm cov nyiaj yog cov nram no hais tias:
- ruaj khov angina;
- vasoconstriction los yog vasospasm;
- vasospastic angina;
- Arterial tawg (raws li monotherapy los yog nyob rau hauv ua ke nrog nrog lwm yam tshuaj);
- nonischemic dilated cardiomyopathy.
Nyob rau hauv tej rooj plaub, cov tshuaj tau "Amlodipine" yuav pom zoo? Nyob rau dab tsi ua rau cov tshuaj no? Nws yog feem ntau tus kws kho nrog rau antianginal tshuaj, xws li cov neeg mob uas yog resistant rau cov kev kho mob ntawm beta-blockers los yog nitrates.
Bans lub txais tos ntawm cov tshuaj
Tam sim no uas koj paub lub hom phiaj uas cov neeg mob yuav tsum tau txais ib tug "Amlodipine" tshuaj. Indications cov tshuaj no uas tau teev tseg saum toj no.
Nrog kev xav txog cov contraindications, siv cov tshuaj no yog txwv tsis pub, yog hais tias hypotension. Nyob rau hauv tas li ntawd, nws tsis pom zoo kom siv ntawm ib tug me nyuam, raws li zoo raws li lub xub ntiag ntawm npau taws me ntsis rau nws cov khoom xyaw.
Yuav ua li cas kuv yuav tsum tau coj cov tshuaj "Amlodipine"?
Analogues, tus nqi ntawm cov tshuaj no muaj li nram no.
Cov kev kawm txhais tau tias yog siv tau rau qhov ncauj thawj coj. Cov tshuaj ntawm cov tshuaj yog xam tus kws kho mob, nyob ntawm seb tus neeg mob tus mob.
Rau cov neeg mob uas kub siab (arterial) thiab angina Tsawg heev koob tshuaj ntawm cov tshuaj ib hnub twg yog 5 mg. Yog hais tias yuav tsum tau, nyob rau hauv cov nram no yog nws ua tau rau kom tus nqi raws nraim ob zaug, uas yog, coj mus txog rau 10 mg ib hnub twg.
Nyob rau hauv cov kev kho mob ntawm dilated cardiomyopathy active medicament yog pom zoo kom noj ib koob tshuaj ntawm 2.5 mg. Yog hais tias zoo taus tshuaj tus nqi yuav muab ntau zog plaub lub sij hawm.
Raws li cov kws txawj, ntau tshaj qhov pom zoo noj tshuaj npaum cas ntawm cov tshuaj (ntau tshaj 10 mg ib hnub twg) yog tsis pom zoo vim qhov no yuav ua tau kom pliaj teebmeem.
Txais tos "amlodipine" nyob rau hauv nrog beta-blockers, diuretics (thiazide) thiab ACE inhibitors tsis yuav tsum tau ntau npaum haum.
Kev nqis tes ua los ntawm-cim
Raws li zam lub txim rau cov tshuaj "Amlodipine"? Sab los ntawm cov tshuaj no yog zoo tsis tuaj kawm ntawv. Txawm li cas los, nyob rau hauv tej rooj plaub (piv txwv li, tsis raws kev cai nrog tus ntau npaum), nws muaj peev xwm tseem ua rau:
- tachycardia, gingival hyperplasia, yaug kais dej, nkees nkees;
- arrhythmia, xeev siab, palpitations, mob taub hau, ua tsis taus pa;
- ntse mob plab, peripheral edema, qaug zog;
- hypotension, tawm pob, paresthesia, pruritus, kiv taub hau.
Nws yuav tsum tau muab sau tseg tias cov mob thawj coj xam tau tias yog ntsiav tshuaj, tus neeg mob tej zaum yuav muaj kev mob nyob rau hauv lub nqua.
Mob ntawm tshuaj overdose
Ntaub ntawv hais txog cov tshuaj overdose mob, cov ntaub ntawv yog tsis muaj hnub no. Txawm tias clinicians hais tias thaum uas tau txais ib tug loj npaum li cas ntawm cov tshuaj nyob rau hauv cov neeg mob tej zaum yuav qhia loj sab tshua.
tshuaj cov kev sib tshuam
Yog nws permissible rau ua ke nrog rau lwm cov tshuaj noj tshuaj "Amlodipine"? Cov lus qhia, cov lus los ntawm cov kws txawj cam hais tias lub hypotensive nyhuv uas cov tshuaj no yog kho kom zoo thaum nws ua ke nrog calcium channel blockers. Ib tug zoo xws li cov tshwm sim yuav tsum los ntawm kev siv txhais tau tias npaj rau nqus tau pa tshuaj loog, thiab orlistat. Incidentally, xws li ib tug ua ke tej zaum yuav txawm ntxias ib tug hypertensive ntsoog.
Txo antigipetrenzivnogo nyhuv thiab sodium tuav nyob rau hauv tib neeg lub cev muaj cai nrog cov ntsiav tshuaj "Amlodimpin" estrogen thiab sympathomimetics.
Cov kev loj hlob ntawm tej tsos mob ntawm neurotoxicity, raws li tinnitus, xeev siab, ataxia, ntuav thiab raws plab, tshwm sim los ntawm lub simultaneous txais tos ntawm amlodipine thiab lithium carbonate.
Tib siv cov tshuaj thiab suav hais tias "Indomethacin", thiab lwm yam narcotics yuav muab thiaj li antihypertensive nyhuv ntawm tus thawj.
Kev pub niam mis thiab cev xeeb tub
Kev Nyab Xeeb ntawm cov tshuaj "Amlodipine" thaum lub sij hawm cev xeeb tub tsis tau kawm. Tib yam siv rau lub sij hawm ntawm lactation. Nyob rau hauv no hais txog, cov hais tias cov khoom nyob rau hauv xws chaw yuav tsum tau siv yog hais tias qhov uas yuav kom tus me nyuam npaum li cas tsawg pab rau cov kev kho mob ntawm cov leej niam.
General tswv yim pom zoo rau lub txais tos ntawm cov tshuaj
Cov kev cai annexed rau cov ntsiav tshuaj, cav hais tias lawv yuav tsum tau noj nrog huab ceev faj nyob rau hauv yuam cai ntawm lub siab thiab ob lub raum, raws li tau zoo raws li aortic stenosis.
Haum ntawm cov tshuaj uas tau raug hais saum toj no, cov neeg laus yuav tsis tau.
Lub medicament "Amlodipine" yuav siv tau rau cov kev kho mob ntawm cov neeg mob nrog paub hais tias raws li dilated cardiomyopathy (nonischemic), uas yog nrog los ntawm lub plawv tsis ua hauj lwm (mob xwm).
Soj ntsuam kev tshawb fawb rau daim ntawv thov ntawm no yeeb tshuaj nyob rau hauv xyuas cov neeg mob tsis tau ua.
Cov ntsiab lus uas muag thiab cia, yuav tsum tau muag
Cia cov tshuaj no yuav tsum muaj nyob rau hauv ib tug maub, qhuav qhov chaw nyob qhov twg qhov kub thiab txias tsis pub tshaj 25 degrees, thiab yog qhov uas tsis muaj kev nkag tau mus rau cov me nyuam yaus.
Tso tawm lub tsev no tsis muaj ib tug kws kho mob tshuaj. Raws li cov kev qhia ntawv, nws cov txee lub neej yog 24 lub hlis. noj cov tshuaj tom qab lub sij hawm ntawm lub sij hawm no yog txwv tsis pub.
Tus nqi ntawm cov tshuaj nyob rau hauv pharmacies thiab zoo sib xws npaj
Yuav ua li cas npaum li cas yog cov "Amlodipine" ntsiav tshuaj? Tus nqi ntawm cov khoom no tej zaum yuav sib txawv, tab sis nyob rau hauv txhua rooj plaub nws tsis yog heev. Tshuaj ntawm ib koob tshuaj ntawm 10 mg nqi txog 55 rubles, thiab nyob ib koob tshuaj 5 mg - txog 35 rubles.
Raws li hais saum toj no, tawg yog ib tug ntau tus kab mob. Yog li ntawd, kws tuam txhab uas muag ua txhua txhua xyoo ntau thiab ntau cov tshuaj tsim los txo cov ntshav siab. Los ntawm txoj kev, tshwj xeeb nyob rau hauv qhia cov cuab yeej, muaj ntau ntau yam. Cov kws kho mob hais tias antihypertensive zog yog cov yam ntxwv ntawm cov nram qab no cov tshuaj: "Agen", "Tenoks", "Akridipin", "Stamlo M", "adipic", "Stamlo", "Amlo", "normodipin" "Amlodipine Sandoz", " Omelar cardio "," Vero Amlodipine, "" Norvasc "" Amlodipine-Teva "," Cordy Cor "," Amlodak "," Norvadin "," Amlovas "," Korvadil "," Amlodigamma "," cardilopin "," amlodipine alkaloid "," Karmagip "," Amlodhi "," Kalchek "" amlodipine Zentiva "," Amlonorm "" amlodipine-Agio "," Amlotop "" amlodipine cardio "," Amlorus "," Amlodifarm "" amlodipine besylate "," Amlong "," Am lokard-Sanovel "thiab t. d.
Posts cov neeg mob thiab cov kws kho mob
Nrog lub hnub nyoog, xws kab mob raws li tawg, yog raug rau ib tug zuj zus tooj ntawm cov neeg. Raws li peb paub, qhov no tshwm sim yog tsiag ntawv los ntawm cov nram qab no cov tsos mob: kiv kiv taub hau, ntev li qaug zog, mob taub hau, tsis muaj zog, darkening ntawm lub qhov muag, koj nkees nkees, thiab tshaj. Raws li kws txawj, tag nrho cov ntawm cov tsos mob ploj nyob rau hauv ib ob peb teev tom qab noj mov "Amlodipine" ntsiav tshuaj nyob rau hauv koob tshuaj ntawm 5 los yog 10 mg.
Cov kws kho mob qhia tias cov tshuaj nyob rau hauv lo lus nug yog ib tug ntawm cov ceev tshaj plaws thiab txhais tau tias zoo. Nyob rau hauv ib tug luv luv lub sij hawm ntawm lub sij hawm nws stabilizes ntshav siab ntawm tus neeg mob, thiab zoo heev pab txoj kev nws mob.
Raws li rau tau txais kev pab, lawv hais tias nws yooj yim txoj kev ntawm daim ntawv thov thiab hauv daim ntawv ntawm qhov cuab tam nrog virtues. Yuav kom txo tau cov ntshav siab, cov neeg mob yuav tsum tau coj ib tug hluas ntsiav tshuaj. Yog li cov kws kho mob ceeb toom hais tias cov tshuaj no overdose yuav ua rau kom los yog txhim khu cov tsos ntawm cov nyom tshua. Nyob rau hauv no hais txog, lawv tsis pom zoo kom siv ntau tshaj 10 mg ntawm cov tshuaj ib hnub twg.
Peb kuj yuav tsum nco ntsoov hais tias ib tug loj pes tsawg tus neeg zoo siab uas tsis muaj nqi ntawm hais tias txhais tau hais tias, raws li tau zoo raws li nws txaus nyob rau hauv tag nrho cov khw muag tshuaj thiab muaj peev xwm mus hloov cov counterparts.
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